SCHEMBL645794

SCHEMBL645794

COc1cc(O)c(-c2nnc(O)n2-c2ccccc2C)cc1C(=O)N(C)Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 12/20 0.58
HSP90AB1 P08238 8/20 0.58
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
KMT2A Q03164 1/20 0.46
HSD17B1 P14061 1/20 0.44
HSD17B2 P37059 1/20 0.44
HTT P42858 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
PDK1 Q15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL644502 0.89 HSP90AA1 (0.71) HSP90AA1HSP90AB1KMT2A
SCHEMBL10170490 0.87 HSP90AA1 (0.65) HSP90AA1HSP90AB1KMT2A
SCHEMBL10170484 0.86 HSP90AA1 (0.58) HSP90AA1HSP90AB1KMT2APDK1
SCHEMBL645220 0.86 HSP90AA1 (0.75) HSP90AA1HSP90AB1KMT2APDK1
SCHEMBL10170483 0.85 HSP90AA1 (0.52) HSP90AA1HSP90AB1GAAHPGDKMT2A
SCHEMBL644590 0.85 HSP90AA1 (0.63) HSP90AA1HSP90AB1HPGDHSD17B2PDK1
SCHEMBL645474 0.84 HSP90AA1 (0.74) HSP90AA1HSP90AB1KMT2APDK1
SCHEMBL645310 0.84 HSP90AA1 (0.64) HSP90AA1HSP90AB1
SCHEMBL646626 0.83 HSP90AA1 (0.62) HSP90AA1HSP90AB1KMT2A
SCHEMBL647220 0.82 HSP90AA1 (0.61) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2023922-B1 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2012-07-11 EP claimed
US-8119795-B2 Triazole derivatives II MERCK PATENT GMBH (DE) 2012-02-21 US claimed
EP-2023922-B1 TRIAZOLE DERIVATIVES II MERCK PATENT GMBH (DE) 2012-07-11 EP disclosed