SCHEMBL6464405

SCHEMBL6464405

Cc1c(C(=O)NC2CCCCC2O)cc(-c2ccc(Cl)cc2Cl)n1CC1CCCCC1

nearest known ligand 0.71

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 15/20 0.71
CNR2 P34972 7/20 0.50
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
TAS1R2 Q8TE23 1/20 0.47
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44
SLC6A4 P31645 2/20 0.44
CHRM1 P11229 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13717726 1.00 CNR1 (0.71) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13602554 1.00 CNR1 (0.71) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13717376 1.00 CNR1 (0.71) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13717141 1.00 CNR1 (0.71) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13717274 0.93 CNR1 (0.79) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13717145 0.93 CNR1 (0.79) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13717212 0.93 CNR1 (0.79) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13602730 0.93 CNR1 (0.69) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL13602643 0.91 CNR1 (0.69) CNR1CNR2TAS1R3TAS1R1TAS1R2
SCHEMBL3922294 0.89 CNR1 (0.56) CNR1CNR2HTR2AHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-10-12 EP disclosed
WO-2004060870-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2004-07-22 WO disclosed