SCHEMBL6464574

SCHEMBL6464574

COc1ccc(CNC(=O)c2ccc3[nH]c(=O)n(C(C)c4ccc(CC(=O)O)cc4)c(=O)c3c2)cc1.O=C(O)C1NCc2ccccc2N1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
MAPT P10636 3/20 0.40
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
ESR1 P03372 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
DRD2 P14416 2/20 0.37
MMP13 P45452 2/20 0.37
USP2 O75604 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
B3GNT2 Q9NY97 1/20 0.36
BRD4 O60885 1/20 0.36
HDAC1 Q13547 1/20 0.36
EPHX2 P34913 1/20 0.36
PPARG P37231 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6235392 0.87 MEN1 (0.54) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL6239501 0.81 MEN1 (0.56) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL6466931 0.80 MEN1 (0.54) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL6218995 0.80 MEN1 (0.54) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL7019551 0.78 PPARG (0.57) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL6237471 0.78 PPARG (0.57) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL6232314 0.77 B3GNT2 (0.46) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL6236358 0.77 MEN1 (0.50) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL6239453 0.77 MEN1 (0.55) MEN1KMT2AMAPTALDH1A1KDM4E
Choline SCHEMBL7021461 0.77 MEN1 (0.49) MEN1KMT2AMAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1530475-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 AND A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 Warner-Lambert Company LLC (US) 2005-05-18 EP disclosed
WO-2004006931-A2 PHARMACEUTICAL COMPOSTIONS COMPRISING AN ALLOSTERIC CARBOXYLIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 AND A SELECTIVE INHIBITOR OF CYCLOOXYGENASE-2 WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed