SCHEMBL6467725

SCHEMBL6467725

COc1cc(C(=O)N2CCCC2c2nc(C)cs2)cc(-c2nnc(C(C)(Cc3ccccc3)NC(=O)OC(C)(C)C)o2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.36
KLK5 Q9Y337 1/20 0.35
TRPV1 Q8NER1 2/20 0.35
CPT1A P50416 5/20 0.34
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
MAPT P10636 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ACE P12821 1/20 0.33
POLB P06746 1/20 0.33
CPT2 P23786 3/20 0.32
CPT1B Q92523 1/20 0.32
KCNQ1 P51787 1/20 0.32
KCNK3 O14649 1/20 0.32
SCD O00767 1/20 0.32
SCD5 Q86SK9 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2727131 0.95 SMN1; SMN2 (0.38) SMN1; SMN2TRPV1CPT1ANPC1RAB9A
SCHEMBL6466775 0.94 ACACB (0.40) SMN1; SMN2KLK5TRPV1CPT1AACACB
SCHEMBL2728516 0.93 SMN1; SMN2 (0.35) SMN1; SMN2KLK5TRPV1ACACBACACA
SCHEMBL6467607 0.92 SMN1; SMN2 (0.37) SMN1; SMN2KLK5TRPV1CPT1AACACB
SCHEMBL6466318 0.92 SMN1; SMN2 (0.37) SMN1; SMN2KLK5TRPV1CPT1AACACB
SCHEMBL6467618 0.92 SMN1; SMN2 (0.37) SMN1; SMN2KLK5TRPV1CPT1AACACB
SCHEMBL6466750 0.92 SMN1; SMN2 (0.37) SMN1; SMN2KLK5TRPV1CPT1AACACB
SCHEMBL2725565 0.92 SMN1; SMN2 (0.34) SMN1; SMN2KLK5TRPV1CPT1AACACB
SCHEMBL2725564 0.92 SMN1; SMN2 (0.34) SMN1; SMN2KLK5TRPV1CPT1AACACB
SCHEMBL2727853 0.91 SMN1; SMN2 (0.36) SMN1; SMN2KLK5TRPV1CPT1AACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed