SCHEMBL6475460

SCHEMBL6475460

O=C(O)c1ccccc1Nc1ccc(CCc2ccc(OCc3ccccc3)cc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 3/20 0.73
CTSV O60911 5/20 0.67
CTSL P07711 5/20 0.67
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
TDP1 Q9NUW8 2/20 0.60
RECQL P46063 1/20 0.60
BLM P54132 1/20 0.60
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
TEAD4 Q15561 1/20 0.55
FFAR1 O14842 1/20 0.55
FFAR4 Q5NUL3 1/20 0.55
FABP4 P15090 1/20 0.52
CHRM4 P08173 1/20 0.52
CHRM3 P20309 1/20 0.52
CLCN2 P51788 1/20 0.52
NR4A1 P22736 1/20 0.51
NR4A2 P43354 1/20 0.51
NR4A3 Q92570 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10833797 0.95 SIRT2 (0.80) SIRT2CTSVCTSLMEN1KMT2A
SCHEMBL6482855 0.88 SIRT2 (0.77) SIRT2CTSVCTSLMEN1KMT2A
SCHEMBL6475801 0.87 MEN1 (0.79) SIRT2CTSVCTSLMEN1KMT2A
SCHEMBL6475772 0.86 MEN1 (0.76) SIRT2CTSVCTSLMEN1KMT2A
SCHEMBL6475426 0.85 MEN1 (0.64) SIRT2CTSVCTSLMEN1KMT2A
SCHEMBL10934405 0.84 SIRT2 (0.76) SIRT2CTSVCTSLMEN1KMT2A
SCHEMBL10833856 0.83 SIRT2 (0.74) SIRT2CTSVCTSLKMT2AALDH1A1
SCHEMBL6482582 0.82 PLK1 (0.64) SIRT2MEN1KMT2ATDP1RECQL
SCHEMBL6484679 0.81 MEN1 (0.57) SIRT2CTSVCTSLMEN1KMT2A
SCHEMBL6475302 0.81 MEN1 (0.54) SIRT2CTSVCTSLMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6972287-B1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits PFIZER INC. (US) 2005-12-06 US claimed
US-20040220235-A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits AUGELLI-SZAFRAN CORINNE ELIZAB (US) 2004-11-04 US claimed
CN-1378446-A Method for inhibiting amyloid aggregation and imaging amyloid deposits WARNER LAMBERT CO (US) 2002-11-06 CN claimed
EP-1225886-A2 METHOD OF INHIBITING AMYLOID PROTEIN AGGREGATION AND IMAGING AMYLOID DEPOSITS WARNER-LAMBERT COMPANY (US) 2002-07-31 EP claimed
WO-2000076489-A2 METHOD OF INHIBITING AMYLOID PROTEIN AGGREGATION AND IMAGING AMYLOID DEPOSITS WARNER-LAMBERT COMPANY (US) 2000-12-21 WO claimed
US-6972287-B1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits PFIZER INC. (US) 2005-12-06 US disclosed
US-20040220235-A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits AUGELLI-SZAFRAN CORINNE ELIZAB (US) 2004-11-04 US disclosed
CN-1378446-A Method for inhibiting amyloid aggregation and imaging amyloid deposits WARNER LAMBERT CO (US) 2002-11-06 CN disclosed
EP-1225886-A2 METHOD OF INHIBITING AMYLOID PROTEIN AGGREGATION AND IMAGING AMYLOID DEPOSITS WARNER-LAMBERT COMPANY (US) 2002-07-31 EP disclosed
WO-2000076489-A2 METHOD OF INHIBITING AMYLOID PROTEIN AGGREGATION AND IMAGING AMYLOID DEPOSITS WARNER-LAMBERT COMPANY (US) 2000-12-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040220235-A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits APP, PSEN1, BACE1 SIRT2 2735/4885CTSV 2743/4885CTSL 3193/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.