SCHEMBL6479290

SCHEMBL6479290

COc1cc(Nc2ncnc(Cl)n2)cc(OCN2CCOCC2)c1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHB4 P54760 3/20 0.50
ZAP70 P43403 1/20 0.46
KDR P35968 2/20 0.46
AURKB Q96GD4 2/20 0.46
IGF1R P08069 2/20 0.45
BRD4 O60885 1/20 0.43
JAK2 O60674 3/20 0.43
JAK3 P52333 2/20 0.43
JAK1 P23458 1/20 0.43
TYK2 P29597 1/20 0.43
FLT3 P36888 2/20 0.43
TBK1 Q9UHD2 2/20 0.43
FYN P06241 2/20 0.43
PTK2 Q05397 5/20 0.42
AURKA O14965 1/20 0.42
DAPK3 O43293 1/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
ABL1 P00519 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6482909 0.90 SRC (0.52) EPHB4ZAP70KDRAURKBIGF1R
SCHEMBL6479263 0.86 SYK (0.57) EPHB4ZAP70KDRJAK3ABL1
SCHEMBL4946510 0.82 EPHB4 (0.69) EPHB4KDRAURKBIGF1RJAK2
SCHEMBL6483193 0.78 KDR (0.57) EPHB4KDRJAK3FLT3DAPK3
SCHEMBL6479597 0.73 KDR (0.57) EPHB4KDRAURKBIGF1RJAK2
SCHEMBL17630988 0.70 FGFR3 (0.53) KDRIGF1RJAK2TBK1FGFR1
SCHEMBL12185363 0.70 ZAP70 (0.73) ZAP70IGF1RJAK2JAK3FLT3
SCHEMBL14214558 0.69 ZAP70 (0.73) ZAP70FLT3TBK1PRKD3LCK
SCHEMBL13325996 0.69 PTK2 (0.62) EPHB4KDRAURKBIGF1RJAK2
SCHEMBL6493240 0.69 KDR (0.56) EPHB4KDRIGF1RJAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6864255-B2 Substituted triazinyl amide derivatives and methods of use AMGEN INC. (US) 2005-03-08 US disclosed
US-20030087908-A1 Substituted triazinyl amide derivatives and methods of use AMGEN INC. 2003-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030087908-A1 Substituted triazinyl amide derivatives and methods of use FLT4, FLT1, VEGFA EPHB4 2420/4885ZAP70 2792/4885KDR 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.