SCHEMBL6482433

SCHEMBL6482433

NC(c1ccc2oc3ccc(F)cc3c2c1)c1ccco1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.35
ALDH1A1 P00352 5/20 0.34
MAPT P10636 5/20 0.34
GABRP O00591 5/20 0.34
GABRD O14764 5/20 0.34
GABRA1 P14867 5/20 0.34
GABRB1 P18505 5/20 0.34
GABRG2 P18507 5/20 0.34
GABRB3 P28472 5/20 0.34
GABRA5 P31644 5/20 0.34
GABRA3 P34903 5/20 0.34
GABRA2 P47869 5/20 0.34
GABRB2 P47870 5/20 0.34
GABRA4 P48169 5/20 0.34
GABRE P78334 5/20 0.34
GABRA6 Q16445 5/20 0.34
GABRG1 Q8N1C3 5/20 0.34
GABRG3 Q99928 5/20 0.34
GABRQ Q9UN88 5/20 0.34
MEN1 O00255 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6483959 0.85 MAPT (0.47) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL6483035 0.77 MEN1 (0.34) TNKSGABRPGABRDGABRA1GABRB1
SCHEMBL6765610 0.77 CYP1A2 (0.44) TNKSALDH1A1MAPTGABRPGABRD
SCHEMBL6485988 0.75 DPP4 (0.38) TNKSALDH1A1GABRPGABRDGABRA1
SCHEMBL6495849 0.75 MAPT (0.37) TNKSALDH1A1MAPTGABRPGABRD
SCHEMBL6482495 0.74 KCNA5 (0.38) ALDH1A1MAPTHPGDPOLBHSD17B10
SCHEMBL6775758 0.74 MAPT (0.37) TNKSALDH1A1MAPTGABRPGABRD
SCHEMBL6495063 0.74 MAPT (0.35) TNKSALDH1A1MAPTGABRPGABRD
SCHEMBL6482835 0.73 MEN1 (0.33) TNKSGABRPGABRDGABRA1GABRB1
SCHEMBL6492261 0.73 CCNC (0.36) TNKSALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050075332-A1 Tricyclic compounds with antiviral activity WARNER LAMBERT COMPANY 2005-04-07 US claimed
US-6800656-B2 Tricyclic compounds and method of treating herpes virus WARNER LAMBERT COMPANY 2004-10-05 US claimed
US-20030229073-A1 Tricyclic compounds and method of treating herpes virus BOOTH RICHARD JOHN (US) 2003-12-11 US claimed
EP-1248777-A2 TRICYCLIC COMPOUNDS WITH ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 2002-10-16 EP claimed
WO-2001051479-A2 TRICYCLIC COMPOUNDS WITH ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 2001-07-19 WO claimed
US-20050075332-A1 Tricyclic compounds with antiviral activity WARNER LAMBERT COMPANY 2005-04-07 US disclosed
US-6800656-B2 Tricyclic compounds and method of treating herpes virus WARNER LAMBERT COMPANY 2004-10-05 US disclosed
US-20030229073-A1 Tricyclic compounds and method of treating herpes virus BOOTH RICHARD JOHN (US) 2003-12-11 US disclosed
EP-1248777-A2 TRICYCLIC COMPOUNDS WITH ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 2002-10-16 EP disclosed
WO-2001051479-A2 TRICYCLIC COMPOUNDS WITH ANTIVIRAL ACTIVITY WARNER-LAMBERT COMPANY (US) 2001-07-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229073-A1 Tricyclic compounds and method of treating herpes virus HDAC8, ZC3HAV1, ZCCHC8 TNKS 3521/4885ALDH1A1 4486/4885MAPT 2337/4885
US-20050075332-A1 Tricyclic compounds with antiviral activity HDAC8, CDK8, ZC3HAV1 TNKS 4075/4885ALDH1A1 4111/4885MAPT 3500/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.