SCHEMBL6484466

SCHEMBL6484466

Cc1cc(C)c(NC(=O)c2cnc(Nc3ccnc(C)c3)s2)c(C)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 16/20 0.66
MAPK14 Q16539 2/20 0.52
RAB9A P51151 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 1/20 0.48
MAPK13 O15264 1/20 0.47
ABL1 P00519 1/20 0.47
EGFR P00533 1/20 0.47
ERBB2 P04626 1/20 0.47
FYN P06241 1/20 0.47
YES1 P07947 1/20 0.47
LYN P07948 1/20 0.47
HCK P08631 1/20 0.47
FGR P09769 1/20 0.47
KIT P10721 1/20 0.47
BCR P11274 1/20 0.47
SRC P12931 1/20 0.47
JAK3 P52333 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18070204 0.86 LCK (0.69) LCKMAPK14RAB9ASMN1; SMN2NPC1
SCHEMBL775200 0.83 LCK (0.65) LCKMAPK14MAPK13ABL1EGFR
SCHEMBL773380 0.83 LCK (0.78) LCKMAPK14RAB9ANPC1MAPK13
SCHEMBL773130 0.81 LCK (0.62) LCKMAPK14RAB9ASMN1; SMN2MAPK13
SCHEMBL775254 0.80 LCK (0.72) LCKMAPK14MAPK13ABL1EGFR
SCHEMBL772868 0.80 LCK (1.00) LCKMAPK14MAPK13ABL1EGFR
SCHEMBL22038674 0.79 LCK (0.69) LCKMAPK14MAPK13ABL1EGFR
SCHEMBL774817 0.79 LCK (0.60) LCKMAPK14RAB9ASMN1; SMN2NPC1
SCHEMBL772252 0.79 LCK (0.76) LCKMAPK14MAPK13ABL1EGFR
SCHEMBL1540058 0.79 LCK (0.74) LCKMAPK14MAPK13EGFRFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6979694-B2 Drugs such as (5-(((2,4,6-Trimethylphenyl)amino)carbonyl)-4-methyl-2-thiazolyl)carbamic acid, 1,1-dimethylethyl ester, used as enzyme inhibitors, for prohylaxis of inflammatory bowel disease; modulation of immunology BRISTOL-MYERS SQUIBB COMPANY (US) 2005-12-27 US disclosed