SCHEMBL6488892

SCHEMBL6488892

Cc1cccc(/C=C\C(=O)N[C@@H](C)c2cccc(Oc3ccncc3)c2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.49
ROCK1 Q13464 10/20 0.44
ROCK2 O75116 6/20 0.44
PRKG1 Q13976 6/20 0.44
PRKACA P17612 6/20 0.44
GSK3A P49840 6/20 0.44
GSK3B P49841 6/20 0.44
PRKX P51817 6/20 0.44
CLK4 Q9HAZ1 5/20 0.44
RPS6KB1 P23443 4/20 0.44
CDK2 P24941 4/20 0.44
AKT2 P31751 4/20 0.44
PRKCD Q05655 4/20 0.44
PRKG2 Q13237 4/20 0.44
PKN2 Q16513 4/20 0.44
HIPK4 Q8NE63 4/20 0.44
SGK2 Q9HBY8 4/20 0.44
RPS6KA5 O75582 3/20 0.44
MAPK1 P28482 3/20 0.44
CDC42BPA Q5VT25 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6488900 1.00 TDP1 (0.49) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6488897 1.00 TDP1 (0.49) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6486443 0.91 TDP1 (0.50) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6486441 0.91 TDP1 (0.50) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6486435 0.91 TDP1 (0.50) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6502176 0.91 TDP1 (0.62) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6502179 0.91 TDP1 (0.62) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6221619 0.89 TDP1 (0.48) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6204160 0.89 TDP1 (0.48) TDP1ROCK1ROCK2PRKG1PRKACA
SCHEMBL6221614 0.89 TDP1 (0.48) TDP1ROCK1ROCK2PRKG1PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900210-B2 Pyridinyl, pyrimidinyl and pyrazinyl amides as potassium channel openers BRISTOL-MYERS SQUIBB COMPANY (US) 2005-05-31 US disclosed