SCHEMBL6497014

SCHEMBL6497014

CSc1ccc(C=CC(=O)N2CCC(C(=O)NC(CC(C)S)C(=O)O)CC2)c(Cl)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGAL P20701 10/20 0.51
ITGB2 P05107 9/20 0.51
ICAM1 P05362 9/20 0.51
CAPN1 P07384 4/20 0.47
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPK1 P28482 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499094 0.93 CAPN1 (0.54) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL6499090 0.93 CAPN1 (0.54) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL8296816 0.90 CAPN1 (0.53) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL6499199 0.90 CAPN1 (0.53) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL6499198 0.90 CAPN1 (0.53) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL6497403 0.88 ITGAL (0.51) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL6497397 0.88 ITGAL (0.51) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL8298602 0.88 ITGAL (0.51) ITGALITGB2ICAM1CAPN1NPC1
SCHEMBL6497008 0.87 ITGB2 (0.50) ITGALITGB2ICAM1CAPN1MEN1
SCHEMBL8297179 0.87 ITGB2 (0.50) ITGALITGB2ICAM1CAPN1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed