SCHEMBL6502124

SCHEMBL6502124

COc1c(N2CCC(C(CC#N)NCC(=O)OC(C)(C)C)C2)c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.66
KDM4E B2RXH2 9/20 0.57
ALDH1A1 P00352 4/20 0.57
HPGD P15428 4/20 0.57
TDP1 Q9NUW8 3/20 0.57
POLB P06746 2/20 0.57
HSD17B10 Q99714 2/20 0.57
PRKD3 O94806 1/20 0.57
ALOX15 P16050 1/20 0.57
OPRM1 P35372 1/20 0.57
CLK2 P49760 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57
LMNA P02545 2/20 0.55
L3MBTL1 Q9Y468 1/20 0.53
NPSR1 Q6W5P4 1/20 0.52
CYP2C19 P33261 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
ATM Q13315 1/20 0.51
TOP1 P11387 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6527983 0.92 KCNH2 (0.66) KCNH2KDM4EALDH1A1HPGDTDP1
SCHEMBL6529075 0.89 KCNH2 (0.72) KCNH2KDM4EALDH1A1HPGDTDP1
SCHEMBL6530889 0.89 KCNH2 (0.72) KCNH2KDM4EALDH1A1HPGDTDP1
SCHEMBL6530890 0.89 KCNH2 (0.72) KCNH2KDM4EALDH1A1HPGDTDP1
SCHEMBL6501764 0.86 KCNH2 (0.65) KCNH2KDM4EALDH1A1HPGDTDP1
SCHEMBL6528763 0.85 KCNH2 (0.81) KCNH2KDM4EALDH1A1HPGDTDP1
SCHEMBL6532431 0.84 KDM4E (0.57) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL6527542 0.83 KCNH2 (0.67) KCNH2KDM4EALDH1A1HPGDTDP1
Hydrochloric Acid SCHEMBL6527471 0.83 KDM4E (0.56) KCNH2KDM4EALDH1A1HPGDPOLB
SCHEMBL6531613 0.83 KCNH2 (0.82) KCNH2KDM4EALDH1A1HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005051381-A1 Substituted urea-octatydroindols as antagonists of melanin concentrating hormone receptor 1 (MCH1R) BIOVITRUM AB (SE) 2005-06-09 WO claimed
WO-2005051381-A1 Substituted urea-octatydroindols as antagonists of melanin concentrating hormone receptor 1 (MCH1R) BIOVITRUM AB (SE) 2005-06-09 WO disclosed
WO-2005049602-A1 QUINOLONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2005-06-02 WO disclosed