SCHEMBL6504749

SCHEMBL6504749

COc1ccc(OC(=O)N(CC(=O)O)Cc2cccc(OCCc3nc(-c4ccco4)oc3C)c2)cc1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 20/20 0.68
PPARG P37231 18/20 0.68
CYP2C9 P11712 8/20 0.67
KCNH2 Q12809 7/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5425806 0.92 PPARA (0.79) PPARAPPARGCYP2C9KCNH2
SCHEMBL13722168 0.87 PPARA (0.88) PPARAPPARGCYP2C9KCNH2
SCHEMBL5437240 0.86 PPARG (0.55) PPARAPPARGCYP2C9KCNH2
SCHEMBL13721830 0.86 PPARA (0.79) PPARAPPARGCYP2C9KCNH2
SCHEMBL13717586 0.84 PPARA (0.80) PPARAPPARGCYP2C9KCNH2
SCHEMBL13721992 0.84 PPARA (0.87) PPARAPPARGCYP2C9KCNH2
SCHEMBL13717524 0.84 PPARA (0.76) PPARAPPARGCYP2C9KCNH2
SCHEMBL13717575 0.84 PPARA (0.88) PPARAPPARGCYP2C9KCNH2
SCHEMBL13717589 0.83 PPARA (0.80) PPARAPPARGCYP2C9KCNH2
SCHEMBL13719596 0.83 PPARA (0.84) PPARAPPARGCYP2C9KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005049589-A2 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF HYPERLIPIDEMIA, DIABETES, OBESITY AND SIMILAR DISEASES CADILA HEALTHCARE LIMITED (IN) 2005-06-02 WO claimed
WO-2005049589-A2 HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF HYPERLIPIDEMIA, DIABETES, OBESITY AND SIMILAR DISEASES CADILA HEALTHCARE LIMITED (IN) 2005-06-02 WO disclosed