SCHEMBL6505478

SCHEMBL6505478

Clc1ccc(Nc2nnc(OCc3cccnc3)c3ccccc23)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 11/20 0.67
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
KDR P35968 12/20 0.53
CSF1R P07333 2/20 0.52
PDGFRB P09619 2/20 0.52
KIT P10721 2/20 0.52
FLT4 P35916 2/20 0.52
CIT O14578 1/20 0.52
EGFR P00533 1/20 0.52
HLA-A P04439 1/20 0.52
RET P07949 1/20 0.52
PDGFRA P16234 1/20 0.52
RPS6KB1 P23443 1/20 0.52
FRK P42685 1/20 0.52
CDK8 P49336 1/20 0.52
DDR1 Q08345 1/20 0.52
STK3 Q13188 1/20 0.52
PTK6 Q13882 1/20 0.52
MAP3K19 Q56UN5 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6494487 0.87 KDR (0.66) FLT1KDRCSF1RPDGFRBKIT
SCHEMBL8204447 0.80 FLT1 (1.00) FLT1MEN1KMT2AKDRCSF1R
SCHEMBL5753555 0.79 FLT1 (0.80) FLT1MEN1KMT2AKDRCSF1R
SCHEMBL1651296 0.78 FLT1 (0.79) FLT1MEN1KMT2AKDRCSF1R
SCHEMBL6482138 0.76 KDR (0.60) FLT1KDRCSF1RPDGFRBKIT
Hydrochloric Acid SCHEMBL6479719 0.75 KDR (0.59) FLT1KDRCSF1RPDGFRBKIT
SCHEMBL6600180 0.75 KDR (0.52) FLT1MEN1KMT2AKDRCSF1R
SCHEMBL6474476 0.74 KDR (0.76) FLT1KDRCSF1RPDGFRBKIT
Hydrochloric Acid SCHEMBL6600046 0.74 KDR (0.51) FLT1MEN1KMT2AKDRCSF1R
SCHEMBL1382851 0.74 FLT1 (0.60) FLT1MEN1KMT2AKDRCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6903101-B1 Substituted pyridazines and fused pyridazines with angiogenesis inhibiting activity BAYER PHARMACEUTICALS CORPORATION (US) 2005-06-07 US claimed
EP-1208096-A1 SUBSTITUTED PYRIDAZINES AND FUSED PYRIDAZINES WITH ANGIOGENESIS INHIBITING ACTIVITY Bayer Corporation (US) 2002-05-29 EP claimed
WO-2001010859-A1 SUBSTITUTED PYRIDAZINES AND FUSED PYRIDAZINES WITH ANGIOGENESIS INHIBITING ACTIVITY BAYER CORPORATION (US) 2001-02-15 WO claimed
US-6903101-B1 Substituted pyridazines and fused pyridazines with angiogenesis inhibiting activity BAYER PHARMACEUTICALS CORPORATION (US) 2005-06-07 US disclosed
EP-1208096-B1 SUBSTITUTED PYRIDAZINES AND FUSED PYRIDAZINES WITH ANGIOGENESIS INHIBITING ACTIVITY BAYER AG (US) 2004-04-28 EP disclosed
EP-1208096-A1 SUBSTITUTED PYRIDAZINES AND FUSED PYRIDAZINES WITH ANGIOGENESIS INHIBITING ACTIVITY Bayer Corporation (US) 2002-05-29 EP disclosed
WO-2001010859-A1 SUBSTITUTED PYRIDAZINES AND FUSED PYRIDAZINES WITH ANGIOGENESIS INHIBITING ACTIVITY BAYER CORPORATION (US) 2001-02-15 WO disclosed