SCHEMBL6506110

SCHEMBL6506110

CSc1ccc(/C=C/C(=O)N2CCC(C(=O)NC(Cc3ccccc3)C(=O)O)CC2)c(Cl)c1Cl

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 5/20 0.56
ITGB2 P05107 6/20 0.53
ICAM1 P05362 6/20 0.53
ITGAL P20701 6/20 0.53
LMNA P02545 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPK1 P28482 1/20 0.46
KMT2A Q03164 1/20 0.45
POLB P06746 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6506117 1.00 CAPN1 (0.56) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL8297323 1.00 CAPN1 (0.56) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL6505573 0.96 CAPN1 (0.51) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL6497573 0.93 ITGB2 (0.48) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL6497576 0.93 ITGB2 (0.48) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL8297275 0.93 CAPN1 (0.54) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL6497111 0.93 CAPN1 (0.54) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL6497116 0.93 CAPN1 (0.54) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL6534061 0.92 CAPN1 (0.48) CAPN1ITGB2ICAM1ITGALLMNA
SCHEMBL8297666 0.92 CAPN1 (0.48) CAPN1ITGB2ICAM1ITGALLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed