SCHEMBL6507663

SCHEMBL6507663

O=C(O)COc1ccnc2cc(C(=O)O)sc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN3B O60391 9/20 0.49
GRIN1 Q05586 9/20 0.49
GRIN2C Q14957 9/20 0.49
KDR P35968 5/20 0.45
FLT1 P17948 3/20 0.45
MET P08581 2/20 0.43
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
CASP1 P29466 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GRIN2D O15399 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
MAP3K8 P41279 1/20 0.38
PPARG P37231 1/20 0.38
CASP7 P55210 1/20 0.38
NCOA2 Q15596 1/20 0.38
NCOA1 Q15788 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22862230 0.86 GRIN3B (0.64) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL22859701 0.82 GRIN3B (0.61) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL22859518 0.79 GRIN3B (0.65) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL22859648 0.75 GRIN3B (0.62) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL22862186 0.75 GRIN3B (0.62) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL22859470 0.74 GRIN3B (0.59) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL29368421 0.74 GRIN3B (0.59) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL22859682 0.74 GRIN3B (0.59) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL199636 0.74 DAO (0.46) GRIN3BGRIN1GRIN2CKDRFLT1
SCHEMBL29998454 0.74 DAO (0.46) GRIN3BGRIN1GRIN2CKDRFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005081960-A2 INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE 1B WYETH (US) 2005-09-09 WO disclosed