SCHEMBL6509133

SCHEMBL6509133

Cc1[nH]nc2c1c(=O)n(CCCN=C(N(C)C)N(C)C)c1ccc(Cl)cc21

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 13/20 0.70
KCNH2 Q12809 2/20 0.44
AURKA O14965 1/20 0.39
KDR P35968 1/20 0.39
AURKB Q96GD4 1/20 0.39
PLK1 P53350 1/20 0.36
RORA P35398 1/20 0.36
RORC P51449 1/20 0.36
NR1H2 P55055 1/20 0.36
RORB Q92753 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6515748 0.85 CHEK1 (0.77) CHEK1KCNH2AURKAKDRAURKB
SCHEMBL6511411 0.85 CHEK1 (0.80) CHEK1KCNH2AURKAKDRAURKB
Hydrochloric Acid SCHEMBL6523110 0.84 CHEK1 (0.76) CHEK1KCNH2AURKAKDRAURKB
SCHEMBL6517703 0.83 CHEK1 (1.00) CHEK1KCNH2AURKAKDRAURKB
Hydrochloric Acid SCHEMBL6507705 0.82 CHEK1 (0.98) CHEK1KCNH2AURKAKDRAURKB
SCHEMBL6518149 0.82 CHEK1 (1.00) CHEK1KCNH2AURKAKDRAURKB
SCHEMBL6513516 0.81 CHEK1 (0.77) CHEK1KCNH2AURKAKDRAURKB
SCHEMBL6515407 0.80 CHEK1 (0.71) CHEK1KCNH2AURKAKDRAURKB
SCHEMBL6515081 0.79 CHEK1 (0.74) CHEK1KCNH2AURKAKDRAURKB
SCHEMBL6511246 0.78 CHEK1 (0.73) CHEK1KCNH2AURKAKDRAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005028474-A2 PYRAZOLOQUINOLINE DERIVATIVES AS CHK-1 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-03-31 WO disclosed