SCHEMBL6509348

SCHEMBL6509348

CCOc1ccc(C(C(=O)O)C(=O)c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
PARP10 Q53GL7 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
PAX8 Q06710 1/20 0.43
ATM Q13315 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PLA2G4B P0C869 1/20 0.43
MAPT P10636 2/20 0.42
AKR1C3 P42330 1/20 0.42
AKR1C2 P52895 1/20 0.42
MAPK1 P28482 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3798330 0.89 GAA (0.43) TDP1PARP10CA12CA1CA2
SCHEMBL6510520 0.85 AKR1C3 (0.53) CA1CA2RAB9APAX8NPSR1
SCHEMBL10585646 0.84 CNR2 (0.51) TDP1PARP10LMNARAB9APAX8
SCHEMBL6532532 0.81 AKR1C3 (0.50) MAPTAKR1C3AKR1C2PTGS2
SCHEMBL3796271 0.81 CA12 (0.44) TDP1CA12CA1CA2CA7
SCHEMBL6510946 0.81 SRC (0.50) AKR1C3AKR1C2ALDH1A1PTGS2
SCHEMBL6511991 0.80 AKR1C3 (0.51) CA12CA1CA2CA9AKR1C3
SCHEMBL6514821 0.80 AKR1C3 (0.51) AKR1C3AKR1C2
SCHEMBL27491723 0.79 CA12 (0.47) TDP1CA12CA1CA2CA7
SCHEMBL3791834 0.79 CA12 (0.53) CA12CA1CA2CA9AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037828-A1 NOVEL INHIBITORS OF DPP-IV, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD. (KR) 2005-04-28 WO claimed
WO-2005051941-A1 THIONE DERIVATIVES, PROCESSES FOR THE PREPARATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME CJ CORPORATION (KR) 2005-06-09 WO disclosed