SCHEMBL6511040

SCHEMBL6511040

CN(C)C(=O)c1ccc(OC(=O)c2ccc(O)c(Cl)c2)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.51
HSP90AB1 P08238 1/20 0.51
SLC6A2 P23975 4/20 0.44
SLC6A4 P31645 4/20 0.44
SLC6A3 Q01959 2/20 0.44
ESRRA P11474 1/20 0.41
NCEH1 Q6PIU2 1/20 0.40
PDK1 Q15118 4/20 0.40
MAPT P10636 1/20 0.39
ERN1 O75460 1/20 0.39
KCNH2 Q12809 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL355700 0.85 HSP90AA1 (0.67) HSP90AA1HSP90AB1PDK1ERN1ALDH1A1
SCHEMBL2649151 0.82 TSHR (0.53) HSP90AA1HSP90AB1MAPTALDH1A1HPGD
SCHEMBL6511037 0.79 HSP90AA1 (0.59) HSP90AA1HSP90AB1PDK1MAPTERN1
SCHEMBL2649764 0.72 TTR (0.48) MAPTHPGDSMN1; SMN2KMT2A
SCHEMBL767829 0.72 KMT2A (0.54) HSP90AA1HSP90AB1MAPTKMT2A
SCHEMBL198849 0.72 CA1 (0.69) HSP90AA1HSP90AB1PDK1MAPTERN1
SCHEMBL30153190 0.72 CA1 (0.69) HSP90AA1HSP90AB1PDK1MAPTERN1
SCHEMBL14531511 0.72 HSP90AA1 (0.46) HSP90AA1HSP90AB1MAPTALDH1A1HPGD
SCHEMBL16741192 0.71 TDP1 (0.60) SLC6A2SLC6A4SLC6A3MAPTSMN1; SMN2
SCHEMBL8756187 0.70 ESR1 (0.47) HSP90AA1HSP90AB1MAPTSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005023762-A1 PYRROLIDINE-2-CARBONITRILE DERIVATIVES AND THEIR USE AS INHIBITORS OF DIPEPTIDYL PEPTIDASE-IV (DPP-IV) ABBOTT LABORATORIES (US) 2005-03-17 WO disclosed