SCHEMBL6513147

SCHEMBL6513147

CCOc1ccc(Br)nc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.49
ADORA1 P30542 1/20 0.49
KDM4E B2RXH2 3/20 0.43
MAPK1 P28482 2/20 0.43
HSD17B10 Q99714 2/20 0.43
HPGD P15428 4/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 3/20 0.39
GRM5 P41594 2/20 0.39
MAPT P10636 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
S1PR1 P21453 4/20 0.38
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
S1PR3 Q99500 1/20 0.37
TSHR P16473 1/20 0.37
DHFR P00374 1/20 0.36
S1PR4 O95977 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16742675 0.81 S1PR4 (0.34) ADORA2AADORA1KDM4EALDH1A1MAPT
SCHEMBL30082515 0.81 S1PR4 (0.34) ADORA2AADORA1KDM4EALDH1A1MAPT
SCHEMBL29364421 0.79 TSHR (0.44) KDM4EHPGDSMN1; SMN2ALDH1A1MAPT
SCHEMBL4573272 0.79 TSHR (0.44) KDM4EHPGDSMN1; SMN2ALDH1A1MAPT
SCHEMBL14290550 0.79 S1PR4 (0.53) KDM4EMAPK1HSD17B10HPGDSMN1; SMN2
SCHEMBL27409803 0.78 TLR8 (0.49) ADORA2AADORA1KDM4EMAPK1HSD17B10
SCHEMBL34466130 0.78 TLR8 (0.49) ADORA2AADORA1KDM4EMAPK1HSD17B10
SCHEMBL3579306 0.77 SMN1; SMN2 (0.44) ADORA2AADORA1KDM4EMAPK1HSD17B10
SCHEMBL12051661 0.77 KDM4E (0.41) ADORA2AADORA1KDM4EMAPK1HSD17B10
SCHEMBL4573187 0.77 KDM4E (0.50) KDM4EMAPK1SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed