SCHEMBL6516027

SCHEMBL6516027

CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)Cc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACE P12821 3/20 0.70
CTSS P25774 7/20 0.65
CTSK P43235 6/20 0.65
CTSB P07858 2/20 0.65
CTSL P07711 1/20 0.65
ATM Q13315 1/20 0.57
AKT1 P31749 1/20 0.57
KLK5 Q9Y337 1/20 0.55
REN P00797 1/20 0.54
PPARA Q07869 2/20 0.54
PPARG P37231 1/20 0.54
APP P05067 1/20 0.53
CA2 P00918 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17688687 0.89 ACE (0.70) ACECTSSCTSKCTSBCTSL
SCHEMBL10536264 0.89 ACE (0.70) ACECTSSCTSKCTSBCTSL
SCHEMBL2603668 0.89 ACE (0.70) ACECTSSCTSKCTSBCTSL
SCHEMBL27839027 0.89 ACE (0.56) ACECTSSCTSKCTSBCTSL
SCHEMBL6332454 0.88 ACE (0.68) ACECTSSCTSKCTSBCTSL
SCHEMBL638877 0.88 ACE (0.68) ACECTSSCTSKCTSBCTSL
SCHEMBL495795 0.88 ACE (0.68) ACECTSSCTSKCTSBCTSL
SCHEMBL21800418 0.88 ACE (0.68) ACECTSSCTSKCTSBCTSL
SCHEMBL495794 0.88 ACE (0.68) ACECTSSCTSKCTSBCTSL
SCHEMBL30193083 0.88 ACE (0.68) ACECTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP disclosed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO disclosed