SCHEMBL6523130

SCHEMBL6523130

Cc1c2c(=O)[nH]c3ccc(OCCCNC(=O)OC(C)(C)C)cc3c2nn1C1CCCCO1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ATR Q13535 5/20 0.44
BRD4 O60885 2/20 0.37
CA12 O43570 4/20 0.37
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
CA9 Q16790 4/20 0.37
F2R P25116 1/20 0.36
PDE3B Q13370 2/20 0.35
PDE3A Q14432 2/20 0.35
DYRK1A Q13627 1/20 0.35
ATRIP Q8WXE1 2/20 0.35
ADRA2C P18825 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529957 0.83 PARP1 (0.37) PDE3BPDE3A
SCHEMBL6508991 0.82 PARP1 (0.44)
SCHEMBL27032631 0.81 ATR (0.47) ATRBRD4CA12CA1CA2
SCHEMBL6510968 0.75 DRD1 (0.33)
SCHEMBL30803398 0.74 ATR (0.42) ATRBRD4
SCHEMBL6511907 0.74 ATR (0.42) ATRBRD4DYRK1A
SCHEMBL6509041 0.74 ATR (0.42) ATRBRD4DYRK1AATRIP
SCHEMBL6509760 0.74 ATR (0.42) ATRBRD4DYRK1AATRIP
SCHEMBL6508889 0.74 ATR (0.42) ATRBRD4DYRK1A
SCHEMBL6511027 0.74 ATR (0.42) ATRBRD4DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050245563-A1 Chk-1 inhibitors MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245563-A1 Chk-1 inhibitors CHKA, CHKB, CHEK1 ATR 717/4885BRD4 874/4885CA12 4451/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.