SCHEMBL6527612

SCHEMBL6527612

COc1c(N2CCC(C(CNC(C)=O)NCCC#N)C2)ccc2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.64
CYP3A4 P08684 1/20 0.45
GSK3B P49841 2/20 0.40
KDM4E B2RXH2 8/20 0.39
ALDH1A1 P00352 4/20 0.39
HPGD P15428 4/20 0.39
POLB P06746 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
HSD17B10 Q99714 2/20 0.39
PRKD3 O94806 1/20 0.39
ALOX15 P16050 1/20 0.39
OPRM1 P35372 1/20 0.39
CLK2 P49760 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
LMNA P02545 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP2C19 P33261 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6529832 0.91 KCNH2 (0.59) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL6527762 0.89 KCNH2 (0.71) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL6507834 0.87 KCNH2 (0.66) KCNH2GSK3BKDM4EALDH1A1HPGD
SCHEMBL6528801 0.85 KCNH2 (0.72) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL6527249 0.84 KCNH2 (0.81) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL5455097 0.82 KCNH2 (0.39) KCNH2
SCHEMBL6504808 0.82 KCNH2 (0.72) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL5456795 0.81 KCNH2 (0.40) KCNH2
SCHEMBL6533246 0.81 KCNH2 (0.59) KCNH2CYP3A4GSK3BKDM4EALDH1A1
SCHEMBL6529113 0.80 KCNH2 (0.65) KCNH2CYP3A4GSK3BKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005049602-A1 QUINOLONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2005-06-02 WO disclosed