SCHEMBL6531344

SCHEMBL6531344

COC(=O)c1c(C)sc2cc(Oc3ccnc4cc(C(=O)N5CCC(OC)C5)sc34)ccc12

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.50
FLT1 P17948 10/20 0.50
MET P08581 3/20 0.44
ADORA3 P0DMS8 2/20 0.37
ADORA2A P29274 2/20 0.37
ADORA2B P29275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240765 1.00 KDR (0.50) KDRFLT1METADORA3ADORA2A
SCHEMBL5241567 0.93 KDR (0.49) KDRFLT1METADORA3ADORA2A
SCHEMBL5243390 0.93 KDR (0.49) KDRFLT1METADORA3ADORA2A
SCHEMBL5244286 0.91 KDR (0.48) KDRFLT1MET
SCHEMBL5242187 0.89 KDR (0.47) KDRFLT1MET
SCHEMBL5243195 0.89 KDR (0.46) KDRFLT1MET
SCHEMBL5241428 0.87 KDR (0.49) KDRFLT1METADORA3ADORA2A
SCHEMBL5242723 0.85 KDR (0.46) KDRFLT1MET
SCHEMBL5241455 0.84 KDR (0.48) KDRFLT1MET
SCHEMBL5240800 0.84 KDR (0.41) KDRFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6869962-B2 Benzofused heterozryl amide derivatives of thienopyridines useful as therapeutic agents, pharmaceutical compositions including the same, and methods for their use AGOURON PHARMACEUTICALS, INC. (US) 2005-03-22 US disclosed