SCHEMBL6531451

SCHEMBL6531451

COCC(C)(C)NCC(=O)N1CCCC1Cc1nnc(-c2ccccc2)o1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.49
HCRTR2 O43614 2/20 0.49
TSPO P30536 1/20 0.49
OPRK1 P41145 1/20 0.49
HTR2B P41595 1/20 0.49
FFAR4 Q5NUL3 1/20 0.49
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
DPP4 P27487 10/20 0.45
DPP7 Q9UHL4 3/20 0.43
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
PKM P14618 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
DPP8 Q6V1X1 2/20 0.42
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6531135 0.90 HCRTR1 (0.51) HCRTR1HCRTR2TSPOOPRK1HTR2B
SCHEMBL6531040 0.84 DPP4 (0.56) RAB9ADPP4DPP7PKML3MBTL1
SCHEMBL28177280 0.79 HCRTR1 (0.58) HCRTR1HCRTR2TSPOOPRK1HTR2B
SCHEMBL1779345 0.79 HCRTR1 (0.58) HCRTR1HCRTR2TSPOOPRK1HTR2B
SCHEMBL1779344 0.79 HCRTR1 (0.58) HCRTR1HCRTR2TSPOOPRK1HTR2B
SCHEMBL6530130 0.78 DPP4 (0.54) DPP4DPP7DPP8
SCHEMBL1778185 0.76 HCRTR2 (0.55) HCRTR1HCRTR2TSPOOPRK1HTR2B
SCHEMBL1778183 0.76 HCRTR2 (0.55) HCRTR1HCRTR2TSPOOPRK1HTR2B
SCHEMBL6531133 0.75 DPP4 (0.71) DPP4DPP7DPP8
SCHEMBL6530309 0.74 DPP4 (0.58) DPP4DPP7DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037828-A1 NOVEL INHIBITORS OF DPP-IV, METHODS OF PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS AN ACTIVE AGENT LG LIFE SCIENCES LTD. (KR) 2005-04-28 WO disclosed