SCHEMBL6532089

SCHEMBL6532089

CN(C)CCCn1c(=O)c2c(S(C)(=O)=O)nn(C3CCCCO3)c2c2cc(Cl)ccc21

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 1/20 0.39
MPO P05164 3/20 0.37
XDH P47989 3/20 0.37
CHEK1 O14757 4/20 0.37
CNR2 P34972 1/20 0.37
CTSK P43235 1/20 0.35
BACE1 P56817 2/20 0.33
MYLK Q15746 1/20 0.32
WEE1 P30291 2/20 0.32
SCARB1 Q8WTV0 1/20 0.32
PARG Q86W56 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6523707 0.88 TOP1 (0.41) TOP1MPOXDHCHEK1CNR2
SCHEMBL6507186 0.72 HTR2C (0.41) TOP1CHEK1CNR2BACE1
SCHEMBL6511094 0.71 CHEK1 (0.41) CHEK1CNR2
SCHEMBL6515376 0.69 MAPT (0.41) CHEK1CNR2
SCHEMBL6514701 0.69 CHEK1 (0.36) TOP1CHEK1CNR2BACE1
SCHEMBL6522000 0.69 CHEK1 (0.41) CHEK1CNR2
SCHEMBL6517699 0.69 ATR (0.39) CHEK1CNR2
SCHEMBL6514903 0.69 HTR2C (0.37) CHEK1CNR2BACE1
Hydrochloric Acid SCHEMBL6530449 0.69 CHEK1 (0.59) TOP1MPOXDHCHEK1WEE1
SCHEMBL6516690 0.68 CHEK1 (0.42) TOP1CHEK1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005028474-A2 PYRAZOLOQUINOLINE DERIVATIVES AS CHK-1 INHIBITORS MILLENNIUM PHARMACEUTICALS, INC. (US) 2005-03-31 WO disclosed