SCHEMBL6533835

SCHEMBL6533835

O=C(Oc1ccnc(NC(=O)C2CCCCO2)c1)c1cccc(Nc2ccccc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.49
TYK2 P29597 1/20 0.49
ACVRL1 P37023 1/20 0.48
PIP5K1C O60331 10/20 0.47
PIK3CA P42336 9/20 0.47
TP53 P04637 2/20 0.46
PIP5K1B O14986 4/20 0.46
PIP5K1A Q99755 4/20 0.46
PIK3CD O00329 3/20 0.46
PDGFRB P09619 3/20 0.46
PIK3CB P42338 3/20 0.46
PI4KA P42356 3/20 0.46
PIK3CG P48736 3/20 0.46
PDK1 Q15118 3/20 0.46
PI4KB Q9UBF8 3/20 0.46
MAPK8 P45983 2/20 0.46
MAPK10 P53779 2/20 0.46
MAPK14 Q16539 2/20 0.46
HPGD P15428 3/20 0.44
NPC1 O15118 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1518883 0.76 MAPK10 (0.72) JAK2TYK2ACVRL1PIP5K1CPIK3CA
SCHEMBL21348455 0.71 NPC1 (0.56) JAK2TYK2TP53MAPK14HPGD
SCHEMBL10537082 0.70 HPGD (0.70) TP53HPGDNPC1POLBRAB9A
SCHEMBL21348452 0.69 JAK2 (0.53) JAK2TYK2MAPK14HPGDNPC1
SCHEMBL16392152 0.68 HPGD (0.56) TP53HPGDNPC1POLBRAB9A
SCHEMBL27638921 0.67 GCK (0.51) JAK2TYK2PIP5K1CPIK3CANPC1
SCHEMBL6509374 0.67 PIP5K1C (0.80) PIP5K1CPIK3CAPIP5K1BPIP5K1APIK3CD
SCHEMBL30642212 0.67 JAK2 (0.64) JAK2TYK2ACVRL1MAPK14HPGD
SCHEMBL3515305 0.66 TYK2 (1.00) JAK2TYK2
SCHEMBL6502898 0.66 PIP5K1C (0.81) PIP5K1CPIK3CAPIP5K1BPIP5K1APIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003123-A1 NOVEL PYRIDINE DERIVATIVES AS JNK SPECIFIC INHIBITORS ASTRAZENECA AB (SE) 2005-01-13 WO disclosed