SCHEMBL6534240

SCHEMBL6534240

Cc1ccc(-c2cc(NCCO)c3ccc(C)cc3n2)cc1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.58
CYP2C19 P33261 1/20 0.49
ACP1 P24666 2/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 2/20 0.47
HTR1A P08908 1/20 0.47
ADRA1D P25100 1/20 0.47
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
SLC2A1 P11166 2/20 0.46
LATS1 O95835 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6534317 0.99 PDE10A (0.57) PDE10ACYP2C19ACP1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL6534187 0.91 SLC2A1 (0.59) PDE10ACYP2C19ACP1KDM4EALDH1A1
SCHEMBL6534262 0.90 ACP1 (0.57) ACP1
Hydrochloric Acid SCHEMBL6534220 0.89 ACP1 (0.56) ACP1
SCHEMBL17372677 0.88 TACR3 (0.58) PDE10AACP1
Hydrochloric Acid SCHEMBL6534345 0.87 PDE10A (0.72) PDE10ACYP2C19ACP1SLC2A1
Hydrochloric Acid SCHEMBL6534337 0.87 TACR3 (0.57) PDE10AACP1
Hydrochloric Acid SCHEMBL6534404 0.81 PDE10A (0.49) PDE10AACP1KDM4EALDH1A1SLC2A1
Hydrochloric Acid SCHEMBL6534405 0.81 PDE10A (0.49) PDE10AACP1KDM4EALDH1A1SLC2A1
SCHEMBL6534482 0.81 TACR3 (0.62) ACP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP claimed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US claimed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP claimed
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US disclosed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP disclosed