SCHEMBL6534512

SCHEMBL6534512

OC(CNC1CCCC1)COc1cc(-c2ccccc2)nc2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.59
MEN1 O00255 3/20 0.59
LMNA P02545 2/20 0.57
ADRB2 P07550 2/20 0.51
POLB P06746 1/20 0.51
HTR1A P08908 5/20 0.50
ADRB1 P08588 1/20 0.49
ABCB1 P08183 2/20 0.48
ACP1 P24666 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6534517 1.00 KMT2A (0.59) KMT2AMEN1LMNAADRB2POLB
Hydrochloric Acid SCHEMBL6534523 0.99 KMT2A (0.59) KMT2AMEN1LMNAADRB2POLB
Hydrochloric Acid SCHEMBL6534521 0.99 KMT2A (0.59) KMT2AMEN1LMNAADRB2POLB
SCHEMBL6534367 0.98 KMT2A (0.56) KMT2AMEN1LMNAADRB2POLB
SCHEMBL6534362 0.98 KMT2A (0.56) KMT2AMEN1LMNAADRB2POLB
Hydrochloric Acid SCHEMBL6534259 0.97 KMT2A (0.56) KMT2AMEN1LMNAADRB2POLB
Hydrochloric Acid SCHEMBL6534254 0.97 KMT2A (0.56) KMT2AMEN1LMNAADRB2POLB
Hydrochloric Acid SCHEMBL6534648 0.95 KMT2A (0.53) KMT2AMEN1LMNAADRB2POLB
Hydrochloric Acid SCHEMBL6534649 0.95 KMT2A (0.53) KMT2AMEN1LMNAADRB2POLB
SCHEMBL6534248 0.82 CYP2D6 (0.62) LMNAADRB2HTR1AADRB1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP claimed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US claimed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP claimed
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US disclosed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP disclosed