SCHEMBL6538604

SCHEMBL6538604

O=C(Nc1ccccc1)Nc1ccc(C[C@@H](CO)NC[C@H](O)COc2ccc(F)cc2)cc1

nearest known ligand 0.86

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 17/20 0.86
ADRB1 P08588 15/20 0.86
ADRB2 P07550 3/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
ALDH1A1 P00352 1/20 0.48
PKM P14618 1/20 0.48
MAPK1 P28482 1/20 0.48
OPRK1 P41145 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6539537 0.93 ADRB3 (0.81) ADRB3ADRB1ADRB2MEN1KMT2A
SCHEMBL6538626 0.93 ADRB3 (1.00) ADRB3ADRB1ADRB2ALDH1A1PKM
Hydrochloric Acid SCHEMBL6538594 0.92 ADRB3 (0.98) ADRB3ADRB1ADRB2
SCHEMBL6538774 0.91 ADRB3 (0.88) ADRB3ADRB1ADRB2
SCHEMBL6538752 0.91 ADRB3 (0.83) ADRB3ADRB1ADRB2MEN1KMT2A
SCHEMBL6538556 0.90 ADRB3 (0.86) ADRB3ADRB1MEN1KMT2A
Trifluoroacetic Acid SCHEMBL6538900 0.87 ADRB3 (0.78) ADRB3ADRB1ADRB2MEN1KMT2A
SCHEMBL6539731 0.87 ADRB3 (1.00) ADRB3ADRB1ADRB2MEN1KMT2A
SCHEMBL7531125 0.86 ADRB3 (0.86) ADRB3ADRB1ADRB2MEN1KMT2A
Trifluoroacetic Acid SCHEMBL6539367 0.85 ADRB3 (0.92) ADRB3ADRB1ADRB2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6826033-B2 BETA 3 ADRENERGIC RECEPTOR AGONISTS; TREATMENT OF POLLAKIURIA, URINARY INCONTINENCE, OBESITY OR DIABETES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-11-30 US disclosed
US-20040037022-A1 Aminoalcohol derivatives ASTELLAS PHARMA INC. (JP) 2004-02-26 US disclosed