SCHEMBL6546007

SCHEMBL6546007

CCNC(=O)N1CCN(C(=O)c2cc(Oc3ccc(NC(=O)Nc4cc(C(C)(C)C)cc(NC(=O)O)c4OC)c4ccccc34)ccn2)CC1CC

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 14/20 0.49
MAPK14 Q16539 13/20 0.49
SRC P12931 12/20 0.49
SYK P43405 12/20 0.49
CXCL8 P10145 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6546701 0.95 GSK3A (0.48) GSK3AMAPK14SRCSYK
SCHEMBL6545669 0.93 SRC (0.56) GSK3AMAPK14SRCSYK
SCHEMBL6546285 0.88 GSK3A (0.51) GSK3AMAPK14SRCSYK
SCHEMBL6546533 0.87 GSK3A (0.49) GSK3AMAPK14SRCSYK
SCHEMBL6546534 0.86 GSK3A (0.57) GSK3AMAPK14SRCSYK
SCHEMBL6547530 0.85 GSK3A (0.53) GSK3AMAPK14SRCSYK
SCHEMBL6546490 0.84 GSK3A (0.55) GSK3AMAPK14SRCSYKCXCL8
SCHEMBL6547025 0.84 GSK3A (0.60) GSK3AMAPK14SRCSYK
SCHEMBL6546644 0.83 GSK3A (0.61) GSK3AMAPK14SRCSYK
SCHEMBL6546739 0.83 GSK3A (0.51) GSK3AMAPK14SRCSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381592-A1 1,4-DISUBSTITUTED BENZO-FUSED COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-01-21 EP disclosed
WO-2002083628-A1 1,4-DISUBSTITUTED BENZO-FUSED COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-10-24 WO disclosed