SCHEMBL6546088

SCHEMBL6546088

CCN(c1ccccc1)c1nccc(Oc2ccc(NC(=O)Nc3cc(C(C)(C)C)cc(NS(C)(=O)=O)c3OC)c3ccccc23)n1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 18/20 0.62
SRC P12931 10/20 0.62
SYK P43405 10/20 0.62
MAPK14 Q16539 10/20 0.62
CYP3A4 P08684 1/20 0.62
CXCL8 P10145 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6545938 0.92 GSK3A (0.65) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL6643809 0.92 MAPK14 (0.55) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL6545585 0.91 MAPK14 (0.64) GSK3ASRCSYKMAPK14
SCHEMBL6545700 0.90 GSK3A (0.55) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL6305196 0.89 MAPK14 (0.75) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL6298580 0.88 GSK3A (0.69) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL6546195 0.87 GSK3A (0.63) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL6643837 0.87 GSK3A (0.67) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL23967439 0.86 GSK3A (0.67) GSK3ASRCSYKMAPK14CYP3A4
SCHEMBL16138970 0.86 GSK3A (0.67) GSK3ASRCSYKMAPK14CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381592-A1 1,4-DISUBSTITUTED BENZO-FUSED COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-01-21 EP claimed
WO-2002083628-A1 1,4-DISUBSTITUTED BENZO-FUSED COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-10-24 WO claimed
EP-1392661-A1 DIARYLUREA DERIVATIVES USEFUL AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-03-03 EP disclosed
EP-1381592-A1 1,4-DISUBSTITUTED BENZO-FUSED COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2004-01-21 EP disclosed
WO-2002092576-A1 DIARYLUREA DERIVATIVES USEFUL AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-11-21 WO disclosed
WO-2002083628-A1 1,4-DISUBSTITUTED BENZO-FUSED COMPOUNDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-10-24 WO disclosed