SCHEMBL6548346

SCHEMBL6548346

C=CCOC(=O)C1=COCC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
ALDH1A1 P00352 3/20 0.41
HSD17B10 Q99714 2/20 0.41
TSHR P16473 1/20 0.41
SNCA P37840 1/20 0.37
RHOA P61586 1/20 0.35
MAPT P10636 3/20 0.35
POLB P06746 1/20 0.35
KDM4E B2RXH2 3/20 0.34
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
HPGD P15428 2/20 0.34
TP53 P04637 1/20 0.34
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
GAA P10253 1/20 0.32
MAPK1 P28482 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3259058 0.81 CYP3A4 (0.50) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL461106 0.75 CYP3A4 (0.52) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL460399 0.71 CYP3A4 (0.47) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL20183947 0.70 CYP3A4 (0.53) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL8602285 0.70 CYP3A4 (0.46) CYP3A4ALDH1A1HSD17B10TSHRSNCA
Acrylic Acid SCHEMBL459310 0.70 CYP3A4 (0.46) CYP3A4ALDH1A1HSD17B10TSHRSNCA
Methacrylic Acid SCHEMBL459214 0.70 CYP3A4 (0.42) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL2050494 0.69 CYP3A4 (0.41) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL8977231 0.69 CYP3A4 (0.41) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL5184261 0.69 CYP3A4 (0.45) CYP3A4ALDH1A1HSD17B10TSHRSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1250330-B1 PROCESS FOR THE PREPARATION OF 3-FUROATE ESTERS AND NOVEL INTERMEDIATE COMPOUNDS EASTMAN CHEM CO (US) 2004-01-07 EP disclosed
EP-1250330-A1 PROCESS FOR THE PREPARATION OF 3-FUROATE ESTERS AND NOVEL INTERMEDIATE COMPOUNDS EASTMAN CHEMICAL COMPANY (US) 2002-10-23 EP disclosed
WO-2001055127-A1 PROCESS FOR THE PREPARATION OF 3-FUROATE ESTERS AND NOVEL INTERMEDIATE COMPOUNDS EASTMAN CHEMICAL COMPANY (US) 2001-08-02 WO disclosed
US-6184394-B1 ALKYL 3-FUROATES FROM 4-ACYL-2,3-DIHYDROFURANS FROM 4-ACYL-2,3-DIHYDRO-FURANS BY HALOGENATING IN THE PRESENCE OF AN ALKANOL FOLLOWED BY CONTACTING WITH A STRONG BASE; DRUGS; ANTINFLAMMATORY AND -FOULING AGENTS EASTMAN CHEMICAL COMPANY 2001-02-06 US disclosed