Ipratropium

Ipratropium

SCHEMBL65495

CC(C)[N+]1(C)[C@@H]2CC[C@@H]1CC(OC(=O)C(CO)c1ccccc1)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CHRM3

The experimentally established mechanism targets of Ipratropium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 known ✓ P20309 6/20 1.00
CHRM2 P08172 7/20 1.00
CHRM5 P08912 6/20 1.00
CHRM1 P11229 6/20 1.00
CHRM4 P08173 5/20 1.00
MEN1 O00255 3/20 1.00
KMT2A Q03164 3/20 1.00
TSHR P16473 2/20 1.00
SMN1; SMN2 Q16637 2/20 0.95
BLM P54132 4/20 0.78
PABPC1 P11940 1/20 0.78
CYP2C19 P33261 1/20 0.77
CYP3A4 P08684 1/20 0.65
CYP2C9 P11712 1/20 0.65
HIF1A Q16665 1/20 0.65
HSD17B10 Q99714 1/20 0.65
HTR2C P28335 2/20 0.63
KDM4E B2RXH2 1/20 0.63
LMNA P02545 1/20 0.63
POLB P06746 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ipratropium SCHEMBL13293462 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL19680109 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL12210779 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL3124 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL14311544 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL19665229 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL7862886 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL15502093 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL19665230 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4
Ipratropium SCHEMBL3125 1.00 CHRM2 (1.00) CHRM2CHRM5CHRM1CHRM3CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5412 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12168024-B2 Use of functionalised chitosan in the treatment of inflammatory/fibrotic pathologies of the respiratory tract and hepatic pathologies GLYCOCORE PHARMA (IT) 2024-12-17 US claimed
US-20240390364-A1 Novel Pyridine Compositions and their use in methods for preventing or treating diseases, disorders and conditions REID CHRISTOPHER BRIAN (US) 2024-11-28 US claimed
US-20240100084-A1 USE OF FUNCTIONALISED CHITOSAN IN THE TREATMENT OF INFLAMMATORY/FIBROTIC PATHOLOGIES OF THE RESPIRATORY TRACT AND HEPATIC PATHOLOGIES GLYCOCORE PHARMA SRL (IT) 2024-03-28 US claimed
US-20240074944-A1 PECVD COATED PHARMACEUTICAL PACKAGING OAKTREE FUND ADMINISTRATION, LLC 2024-03-07 US claimed
EP-4326283-A1 USE OF FUNCTIONALISED CHITOSAN IN THE TREATMENT OF INFLAMMATORY/FIBROTIC PATHOLOGIES OF THE RESPIRATORY TRACT AND HEPATIC PATHOLOGIES GLYCOCORE PHARMA S.r.l. (IT) 2024-02-28 EP claimed
CN-117241773-A Polymer medicine bottle with standard external dimensions and reduced internal volume SIO2医疗产品有限公司 2023-12-15 CN claimed
EP-4259153-A1 NOVEL USE OF PYRROLOPYRIDINE DERIVATIVES FOR PREVENTING OR TREATING INFLAMMATORY DISEASES Voronoi Inc. (KR) 2023-10-18 EP claimed
US-20230303305-A1 METHOD AND PACKAGE FOR REDUCING THE DEGRADATION OF A DRUG AND/OR EXCIPIENT, E.G. POLYSORBATE STABILIZER, IN A PHARMACEUTICAL PRODUCT OAKTREE FUND ADMINISTRATION, LLC 2023-09-28 US claimed
EP-4247316-A1 POLYMER VIALS HAVING STANDARD EXTERNAL DIMENSIONS AND REDUCED INTERNAL VOLUME SiO2 Medical Products, Inc. (US) 2023-09-27 EP claimed
US-20230277415-A1 POLYMER VIALS HAVING STANDARD EXTERNAL DIMENSIONS AND REDUCED INTERNAL VOLUME SIO2 MEDICAL PRODUCTS, INC. 2023-09-07 US claimed
EP-1058657-A1 CONTAINER FOR A MEDICINAL LIQUID Boehringer Ingelheim International GmbH (DE) 2000-12-13 EP claimed
WO-2000049988-A2 CARTRIDGE FOR A LIQUID BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2000-08-31 WO claimed
CN-1253508-A Topical nasal anti-inflammatory composition WARNER LAMBERT CO (US) 2000-05-17 CN claimed
CN-1240347-A New aqueous medicament preparations for the production of propellent gas-free aerosols BOEHRINGER INGELHELM KG (DE) 2000-01-05 CN claimed
EP-0946146-A2 NEW AQUEOUS MEDICAMENT PREPARATIONS FOR THE PRODUCTION OF PROPELLENT GAS-FREE AEROSOLS Boehringer Ingelheim Pharma KG (DE) 1999-10-06 EP claimed
WO-1999043571-A1 CONTAINER FOR A MEDICINAL LIQUID BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 1999-09-02 WO claimed
WO-1998052580-A1 TREATING ASTHMA BY PREVENTING AND/OR ACCOMMODATING FOR S-NITROSOTHIOL BREAKDOWN DUKE UNIVERSITY (US) 1998-11-26 WO claimed
EP-0853501-A1 DEVICE OF MINIATURISED CONSTRUCTION FOR PRODUCING HIGH PRESSURE IN A FLUID TO BE ATOMISED BOEHRINGER INGELHEIM INTERNATIONAL GmbH (DE) 1998-07-22 EP claimed
WO-1998027959-A2 NEW AQUEOUS MEDICAMENT PREPARATIONS FOR THE PRODUCTION OF PROPELLENT GAS-FREE AEROSOLS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-07-02 WO claimed
WO-1997012687-A1 DEVICE OF MINIATURISED CONSTRUCTION FOR PRODUCING HIGH PRESSURE IN A FLUID TO BE ATOMISED BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 1997-04-10 WO claimed