SCHEMBL6554606

SCHEMBL6554606

CC(C)S(=O)(=O)NC1CCCC1c1ccc(Br)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 13/20 1.00
GRIA2 P42262 8/20 1.00
KCNH2 Q12809 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605805 1.00 GRIA4 (1.00) GRIA4GRIA2KCNH2
SCHEMBL4607668 1.00 GRIA4 (1.00) GRIA4GRIA2KCNH2
SCHEMBL4608168 1.00 GRIA4 (1.00) GRIA4GRIA2KCNH2
SCHEMBL4607332 0.87 GRIA4 (1.00) GRIA4GRIA2KCNH2
SCHEMBL4608724 0.86 GRIA4 (1.00) GRIA4GRIA2KCNH2
SCHEMBL4607921 0.86 GRIA4 (0.77) GRIA4GRIA2KCNH2
SCHEMBL4606591 0.86 GRIA4 (1.00) GRIA4GRIA2KCNH2
SCHEMBL14141323 0.86 GRIA4 (0.77) GRIA4GRIA2KCNH2
SCHEMBL4607609 0.86 GRIA4 (1.00) GRIA4GRIA2KCNH2
SCHEMBL14141331 0.86 GRIA4 (0.77) GRIA4GRIA2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1390072-A2 USE OF AN AMPA RECEPTOR POTENTIATOR FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF TYPE 2 DIABETES ELI LILLY AND COMPANY (US) 2004-02-25 EP disclosed
WO-2002089848-A2 USE OF AN AMPA RECEPTOR POTENTIATOR FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF TYPE 2 DIABETES ELI LILLY AND COMPANY (US) 2002-11-14 WO disclosed