SCHEMBL6556315

SCHEMBL6556315

CCc1c(OC)cc2c(c1OC)C(=O)CC1CN(C)CC21

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.43
ACHE P22303 3/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PTGS2 P35354 1/20 0.31
MKNK2 Q9HBH9 1/20 0.31
TAS2R31 P59538 1/20 0.31
HTT P42858 1/20 0.31
CYP3A4 P08684 1/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6556309 1.00 IDO1 (0.43) IDO1ACHEALDH1A1KDM4ESMN1; SMN2
SCHEMBL6556312 1.00 IDO1 (0.43) IDO1ACHEALDH1A1KDM4ESMN1; SMN2
SCHEMBL6556331 0.90 IDO1 (0.41) IDO1ACHECYP3A4HTR2C
SCHEMBL6556322 0.90 IDO1 (0.41) IDO1ACHECYP3A4HTR2C
SCHEMBL6556326 0.90 IDO1 (0.41) IDO1ACHECYP3A4HTR2C
SCHEMBL13213819 0.90 IDO1 (0.41) IDO1ACHECYP3A4HTR2C
SCHEMBL6556422 0.87 IDO1 (0.58) IDO1ALDH1A1KDM4ESMN1; SMN2PTGS2
SCHEMBL6556426 0.87 IDO1 (0.58) IDO1ALDH1A1KDM4ESMN1; SMN2PTGS2
SCHEMBL6556416 0.87 IDO1 (0.58) IDO1ALDH1A1KDM4ESMN1; SMN2PTGS2
Fumaric Acid SCHEMBL6556498 0.81 IDO1 (0.52) IDO1ALDH1A1KDM4ESMN1; SMN2PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6310208-B1 Serotonin receptor binding benzo[e]isoindoles and benzo[h]isoquinolines HOFFMANN-LA ROCHE INC. 2001-10-30 US claimed
EP-0958285-B1 TRICYCLIC BENZO[e]ISOINDOLES AND BENZO[h]ISOQUINOLINES HOFFMANN LA ROCHE (CH) 2004-01-07 EP disclosed
US-6310208-B1 Serotonin receptor binding benzo[e]isoindoles and benzo[h]isoquinolines HOFFMANN-LA ROCHE INC. 2001-10-30 US disclosed
EP-0958285-A1 TRICYCLIC BENZO[e]ISOINDOLES AND BENZO[h]ISOQUINOLINES F.HOFFMANN-LA ROCHE AG (CH) 1999-11-24 EP disclosed
WO-1998030546-A1 TRICYCLIC BENZO[e]ISOINDOLES AND BENZO[h]ISOQUINOLINES F. HOFFMANN-LA ROCHE AG (CH) 1998-07-16 WO disclosed