SCHEMBL6558159

SCHEMBL6558159

O=CCn1c(-c2ccc(F)cc2)ncc(NC(=O)OCc2ccccc2)c1=O

nearest known ligand 0.63

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ELANE P08246 19/20 0.63
MGLL Q99685 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6085892 0.93 ELANE (0.60) ELANE
SCHEMBL7300356 0.92 ELANE (0.61) ELANE
SCHEMBL6558401 0.91 ELANE (0.56) ELANE
SCHEMBL6556223 0.90 ELANE (0.62) ELANE
SCHEMBL6557626 0.89 ELANE (0.54) ELANE
SCHEMBL6558418 0.89 ELANE (0.64) ELANE
SCHEMBL6557728 0.88 ELANE (0.70) ELANEMGLL
SCHEMBL6556126 0.87 ELANE (0.65) ELANE
SCHEMBL6558347 0.86 ELANE (0.58) ELANEMGLL
SCHEMBL6558341 0.86 ELANE (0.62) ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1188401-C Heterocyclic amide compound and its pharmaceutical use MITSUBISHI PHARMACEUTICAL CO L (JP) 2005-02-09 CN disclosed
EP-0826671-B1 HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USE OF THE SAME MITSUBISHI PHARMA CORP (JP) 2004-12-29 EP disclosed
CN-1131210-C Heterocyclic amide compound and medical use thereof MITSUBISHI SEIYAKU CO LTD (JP) 2003-12-17 CN disclosed
US-6528514-B1 Pyrimidin-4-one-5-amino-3-alkylcarboxamidomethyl compounds WELFIDE CORPORATION (JP) 2003-03-04 US disclosed
CN-1304931-A Heterocyclic amide compound and medical use thereof EFUKU CO LTD (JP) 2001-07-25 CN disclosed
EP-1062949-A1 IgE ANTIBODY PRODUCTION INHIBITORS AND AUTOIMMUNE DISEASES INHIBITORS Welfide Corporation (JP) 2000-12-27 EP disclosed
EP-0528633-B1 Pyrimidinyl acetamides as elastase inhibitors ZENECA LTD (GB) 2000-10-18 EP disclosed
US-6080738-A USEFUL AS CHYMASE INHIBITORS AND CAN BE USED FOR THE PROPHYLAXIS AND TREATMENT OF VARIOUS DISEASES CAUSED BY CHYMASE, SUCH AS THOSE CAUSED BY ANGIOTENSIN II YOSHITOMI PHARMACEUTICALS INDUSTRIES, LTD. (JP) 2000-06-27 US disclosed
EP-0940400-A1 NOVEL HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USES THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1999-09-08 EP disclosed
US-5948785-A USEFUL AS CHYMASE INHIBITORS AND CAN BE EFFECTIVE FOR THE PROPHYLAXIS AND TREATMENT OF VARIOUS DISEASES CAUSED BY CHYMASE, SUCH AS THOSE CAUSED BY ANGIOTENSIN II. THE GREEN CROSS CORPORATION (JP) 1999-09-07 US disclosed
CN-1188472-A Heterocyclic amide compound and medical use thereof GREEN CROSS CORP (JP) 1998-07-22 CN disclosed
US-5736535-A 1-pyrimidinylacetamide compounds which are inhibitors of human leukocyte elastase ZENECA LIMITED (GB) 1998-04-07 US disclosed
EP-0826671-A1 HETEROCYCLIC AMIDE COMPOUNDS AND MEDICINAL USE OF THE SAME THE GREEN CROSS CORPORATION (JP) 1998-03-04 EP disclosed
EP-0636143-B1 ALPHA-AMINOBORONIC ACID PEPTIDES AND THEIR USE AS ELASTASE INHIBITORS ZENECA LTD (GB) 1997-09-24 EP disclosed
EP-0636143-A1 ALPHA-AMINOBORONIC ACID PEPTIDES AND THEIR USE AS ELASTASE INHIBITORS. ZENECA LTD (GB) 1995-02-01 EP disclosed
WO-1993021214-A1 ALPHA-AMINOBORONIC ACID PEPTIDES AND THEIR USE AS ELASTASE INHIBITORS ZENECA LIMITED (GB) 1993-10-28 WO disclosed
US-5254558-A Substituted 1,3-diazines as leukocyte elastase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-19 US disclosed
EP-0528633-A1 Pyrimidinyl acetamides as elastase inhibitors ZENECA LIMITED (GB) 1993-02-24 EP disclosed