SCHEMBL6560101

SCHEMBL6560101

CCCc1cc(CC(=O)O)ccc1OCCCOc1ccc2c(-c3ccccc3)coc2c1CCC

nearest known ligand 0.71

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 19/20 0.71
PPARG P37231 18/20 0.71
PPARA Q07869 17/20 0.71
NR1H2 P55055 4/20 0.52
NR1H3 Q13133 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6559896 0.92 PPARG (0.61) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL6559945 0.89 PPARG (0.84) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL6560081 0.89 PPARA (0.71) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL6560008 0.89 PPARG (0.70) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL6559284 0.86 PPARG (0.72) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL2066214 0.84 PPARG (0.77) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL5973012 0.84 PPARD (0.63) PPARDPPARGPPARANR1H2NR1H3
Toluene SCHEMBL6559134 0.84 PPARG (0.54) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL6560654 0.84 PPARD (0.66) PPARDPPARGPPARANR1H2NR1H3
SCHEMBL5973876 0.83 PPARG (0.63) PPARDPPARGPPARANR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0904079-B1 ANTIDIABETIC AGENTS MERCK & CO INC (US) 2004-03-24 EP disclosed
EP-0904079-A4 1999-05-06 EP disclosed
EP-0904079-A1 ANTIDIABETIC AGENTS Merck & Co., Inc. (US) 1999-03-31 EP disclosed
US-5859051-A ACETYLPHENOL DERIVATIVES MERCK & CO., INC. (US) 1999-01-12 US disclosed
WO-1997027857-A1 ANTIDIABETIC AGENTS MERCK & CO., INC. (US) 1997-08-07 WO disclosed