SCHEMBL6563747

SCHEMBL6563747

NC(=O)C#Cc1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.51
CA2 P00918 3/20 0.51
CA9 Q16790 3/20 0.51
CA1 P00915 2/20 0.51
GFER P55789 1/20 0.50
PARP1 P09874 1/20 0.48
IKBKB O14920 1/20 0.48
GRM5 P41594 5/20 0.45
KCNN4 O15554 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2636049 0.83 GFER (0.55) CA12CA2CA9CA1GFER
SCHEMBL28501126 0.79 GFER (0.48) CA12CA2CA9CA1GFER
SCHEMBL29961896 0.79 GFER (0.48) CA12CA2CA9CA1GFER
SCHEMBL7158136 0.78 NPSR1 (0.39) CA12CA2CA9CA1GFER
SCHEMBL1751529 0.77 GFER (0.50) CA12CA2CA9CA1GFER
SCHEMBL30055201 0.77 HSP90AA1 (0.60) CA12CA2CA9CA1GFER
SCHEMBL27167261 0.77 HSP90AA1 (0.60) CA12CA2CA9CA1GFER
SCHEMBL28909500 0.77 GFER (0.47) CA12CA2CA9CA1GFER
SCHEMBL29941936 0.77 GFER (0.47) CA12CA2CA9CA1GFER
SCHEMBL667669 0.77 GFER (0.57) CA12CA2CA9CA1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944581-A4 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES LILLY CO ELI (US) 2004-09-08 EP disclosed
US-6069247-A REACTING AN ACETYLENECARBOXY AMIDE AND AN ARYL OR HETEROCYCLYL HALIDE OR A GROUP ENHANCING THE ELECTROPHILICITY OF THE ATOM TO WHICH IT IS ATTACHED FOR DISPLACEMENT; USING A PALLADIUM COMPOUND CATALYST, A BASE AND AN ACID ELI LILLY AND COMPANY (US) 2000-05-30 US disclosed
EP-0944581-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1999-09-29 EP disclosed
US-5917038-A REACTING PROPIOLAMIDE WITH ACTIVATED AROMATIC RING IN THE PRESENCE OF A PALLADIUM CATALYST ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed
WO-1998022429-A1 PROCESS OF PREPARING SUBSTITUTED ACRYLAMIDES ELI LILLY AND COMPANY (US) 1998-05-28 WO disclosed