SCHEMBL6564972

SCHEMBL6564972

CC(C)S(=O)(=O)NCC(C)(O)c1ccc(C(C)(O)CNS(=O)(=O)C(C)C)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GRIA4 P48058 7/20 0.41
CYP2C19 P33261 1/20 0.39
EPHX2 P34913 3/20 0.33
NR1H4 Q96RI1 2/20 0.33
GRIA2 P42262 1/20 0.33
TRPV1 Q8NER1 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6563345 0.83 CYP2C19 (0.53) GRIA4CYP2C19EPHX2NR1H4GRIA2
SCHEMBL6564976 0.81 CYP2C19 (0.38) GRIA4CYP2C19HDAC3HDAC1HDAC2
SCHEMBL6565067 0.80 GRIA4 (0.42) GRIA4EPHX2NR1H4GRIA2TRPV1
SCHEMBL13256290 0.79 CYP2C19 (0.49) GRIA4CYP2C19GRIA2
SCHEMBL13255837 0.79 CYP2C19 (0.49) GRIA4CYP2C19GRIA2
SCHEMBL5187414 0.78 CYP2C19 (0.41) GRIA4CYP2C19GRIA2
SCHEMBL14394435 0.77 CYP2C19 (0.48) GRIA4CYP2C19EPHX2NR1H4
SCHEMBL5188496 0.77 CYP2C19 (0.48) GRIA4CYP2C19
SCHEMBL5188470 0.76 GRIA4 (0.48) GRIA4CYP2C19EPHX2
SCHEMBL3703932 0.76 CYP2C19 (0.47) GRIA4CYP2C19EPHX2NR1H4GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296945-B1 SULFONAMIDE DERIVATIVES LILLY CO ELI (US) 2004-08-04 EP disclosed
US-6703425-B2 ADMINISTERING GLUTAMATE RECEPTOR POTENTIATOR TO TREAT PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY 2004-03-09 US disclosed
US-20030229102-A1 Sulfonamide derivatives ELI LILLY AND COMPANY 2003-12-11 US disclosed
EP-1296945-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2003-04-02 EP disclosed
WO-2001096289-A1 SULFONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229102-A1 Sulfonamide derivatives GRIN1, GRIN2A, SLC1A2 GRIA4 17/4885CYP2C19 2069/4885EPHX2 1613/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.