SCHEMBL6565724

SCHEMBL6565724

O=C(c1ccc(OCCN2CCCCC2)cc1)c1c(-c2ccc(OCSc3ccccc3)cc2)sc2cc(OCSc3ccccc3)ccc12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 20/20 0.73
ESR2 Q92731 19/20 0.73
MEN1 O00255 2/20 0.69
ALDH1A1 P00352 2/20 0.69
LMNA P02545 2/20 0.69
TP53 P04637 2/20 0.69
CYP3A4 P08684 2/20 0.69
MAPT P10636 2/20 0.69
ALOX15 P16050 2/20 0.69
KMT2A Q03164 2/20 0.69
HSD17B10 Q99714 2/20 0.69
TDP1 Q9NUW8 2/20 0.69
PLD2 O14939 1/20 0.69
KDM1A O60341 1/20 0.69
NR1I2 O75469 1/20 0.69
USP2 O75604 1/20 0.69
C5 P01031 1/20 0.69
FYN P06241 1/20 0.69
PGR P06401 1/20 0.69
ADRA2A P08913 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6566930 0.89 ESR1 (0.80) ESR1ESR2MEN1ALDH1A1LMNA
Hydrochloric Acid SCHEMBL6565691 0.88 ESR1 (0.80) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL6662322 0.87 ESR1 (0.79) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL11551601 0.86 ESR1 (0.75) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL5166092 0.85 ESR1 (0.76) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL11549535 0.85 ESR1 (0.78) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL8598366 0.85 ESR1 (0.89) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL8598353 0.85 ESR1 (0.89) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL11209650 0.85 ESR1 (0.82) ESR1ESR2MEN1ALDH1A1LMNA
SCHEMBL5225075 0.85 ESR1 (0.84) ESR1ESR2MEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025098-B1 BENZOTHIOPHENES LILLY CO ELI (US) 2004-03-31 EP claimed
US-6403614-B1 SUCH AS 2-(4-(METHYLTHIOMETHOXY)PHENYL)-3-(4-(2-PIPERIDIN-1-YL)ETHOXY) BENZOYL)-6-METHYLTHIOMETHOXYBENZO(B)THIOPHENE;INHIBITION OF OSTEOPOROSIS, HYPERLIPEDEMIA, CANCER, POSTMENOPAUSAL SYNDROME, ELI LILLY AND COMPANY 2002-06-11 US claimed
US-6403614-B1 SUCH AS 2-(4-(METHYLTHIOMETHOXY)PHENYL)-3-(4-(2-PIPERIDIN-1-YL)ETHOXY) BENZOYL)-6-METHYLTHIOMETHOXYBENZO(B)THIOPHENE;INHIBITION OF OSTEOPOROSIS, HYPERLIPEDEMIA, CANCER, POSTMENOPAUSAL SYNDROME, ELI LILLY AND COMPANY 2002-06-11 US disclosed