SCHEMBL6567278

SCHEMBL6567278

COc1ccc(NC(=O)NC23CC4CC(CC(C4)C2)C3)cc1Cl

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 17/20 0.70
MAPT P10636 3/20 0.59
NPSR1 Q6W5P4 3/20 0.59
ALDH1A1 P00352 1/20 0.59
HPGD P15428 1/20 0.59
LMNA P02545 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6566881 0.86 EPHX2 (0.72) EPHX2MAPTNPSR1ALDH1A1HPGD
SCHEMBL4346744 0.82 EPHX2 (1.00) EPHX2MAPTLMNA
SCHEMBL4113279 0.78 EPHX2 (0.65) EPHX2MAPTNPSR1ALDH1A1HPGD
SCHEMBL4348906 0.78 EPHX2 (0.73) EPHX2MAPTNPSR1LMNA
SCHEMBL12932434 0.77 EPHX2 (1.00) EPHX2MAPTALDH1A1
SCHEMBL28399545 0.76 MAPT (0.78) EPHX2MAPTNPSR1LMNA
SCHEMBL6649644 0.76 EPHX2 (0.58) EPHX2MAPTNPSR1ALDH1A1HPGD
SCHEMBL11685462 0.76 SMN1; SMN2 (0.63) MAPTNPSR1ALDH1A1HPGDLMNA
SCHEMBL11754054 0.76 SMN1; SMN2 (0.63) MAPTNPSR1ALDH1A1HPGDLMNA
SCHEMBL15335335 0.76 EPHX2 (1.00) EPHX2MAPTNPSR1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1402887-A1 New compounds for the inhibition of undesired cell proliferation and use thereof Jerini AG (DE) 2004-03-31 EP claimed
EP-1402888-A1 The use of substituted carbocyclic compounds as rotamases inhibitors Jerini AG (DE) 2004-03-31 EP claimed