SCHEMBL6576725

SCHEMBL6576725

O[C@@H]1[C@H](O)[C@@H](c2nnc(C3CCCC3)o2)O[C@H]1n1cnc2c(N[C@@H]3CCC[C@H]3F)ncnc21

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 7/20 0.54
ADORA3 P0DMS8 6/20 0.54
ADORA2A P29274 5/20 0.54
ADORA2B P29275 4/20 0.54
CYP2D6 P10635 1/20 0.54
TSHR P16473 2/20 0.50
PMP22 Q01453 2/20 0.50
GAA P10253 1/20 0.50
HTT P42858 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
SLC29A1 Q99808 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
TP53 P04637 1/20 0.50
NFKB1 P19838 1/20 0.50
HIF1A Q16665 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6576651 0.92 ADORA1 (0.65) ADORA1ADORA3ADORA2AADORA2BCYP2D6
SCHEMBL6576683 0.88 ADORA2A (0.64) ADORA1ADORA3ADORA2AADORA2BTSHR
SCHEMBL6575267 0.87 ADORA1 (0.52) ADORA1ADORA3ADORA2AADORA2BCYP2D6
SCHEMBL6573802 0.87 ADORA2A (0.64) ADORA1ADORA3ADORA2AADORA2BTSHR
SCHEMBL6576742 0.83 ADORA1 (0.53) ADORA1ADORA3ADORA2AADORA2BCYP2D6
SCHEMBL6797276 0.82 ADORA2A (0.65) ADORA1ADORA3ADORA2AADORA2BCYP2D6
SCHEMBL6574622 0.82 ADORA2A (0.65) ADORA1ADORA3ADORA2AADORA2BCYP2D6
SCHEMBL6574707 0.81 ADORA2A (0.64) ADORA1ADORA3ADORA2AADORA2BTSHR
SCHEMBL6575097 0.81 ADORA1 (0.64) ADORA1ADORA3ADORA2AADORA2BCYP2D6
SCHEMBL6572783 0.79 ADORA2A (0.61) ADORA1ADORA3ADORA2AADORA2BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1090019-B1 ADENOSINE DERIVATIVES GLAXO GROUP LTD (GB) 2004-09-29 EP disclosed
EP-1447407-A1 Adenosine derivatives GLAXO GROUP LIMITED (GB) 2004-08-18 EP disclosed