SCHEMBL6578503

SCHEMBL6578503

COc1ccc(-c2nc(-c3cccc(CN4CCCC4)c3)n[nH]2)cc1F

nearest known ligand 0.62

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.62
ADORA1 P30542 2/20 0.62
CNR1 P21554 4/20 0.49
CNR2 P34972 4/20 0.49
S1PR1 P21453 1/20 0.47
KMT2A Q03164 1/20 0.44
DRD4 P21917 4/20 0.43
NR1H2 P55055 1/20 0.42
NR1H3 Q13133 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
HTR7 P34969 1/20 0.41
LCK P06239 1/20 0.41
BTK Q06187 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6582961 0.99 ADORA2A (0.61) ADORA2AADORA1CNR1CNR2S1PR1
Hydrochloric Acid SCHEMBL6580754 0.91 ADORA2A (0.66) ADORA2AADORA1CNR1CNR2S1PR1
SCHEMBL6578583 0.88 ADORA2A (0.62) ADORA2AADORA1CNR1CNR2S1PR1
Hydrochloric Acid SCHEMBL6583845 0.87 ADORA2A (0.61) ADORA2AADORA1CNR1CNR2S1PR1
Hydrochloric Acid SCHEMBL6580863 0.87 ADORA2A (0.61) ADORA2AADORA1CNR1CNR2S1PR1
Hydrochloric Acid SCHEMBL6578773 0.87 ADORA2A (0.58) ADORA2AADORA1CNR1CNR2S1PR1
Hydrochloric Acid SCHEMBL6584484 0.87 ADORA2A (0.68) ADORA2AADORA1CNR1CNR2S1PR1
Hydrochloric Acid SCHEMBL6580955 0.85 ADORA2A (0.61) ADORA2AADORA1CNR1CNR2S1PR1
Hydrochloric Acid SCHEMBL6578211 0.85 ADORA2A (0.58) ADORA2AADORA1S1PR1KMT2ADRD4
SCHEMBL6583869 0.85 ADORA2A (0.65) ADORA2AADORA1CNR1CNR2S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US claimed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP claimed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed