SCHEMBL6579536

SCHEMBL6579536

CCCCCCCCOc1c(O)c2ccc(NC(=O)c3ccccc3)cc2n(C)c1=O

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 4/20 0.48
TP53 P04637 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7997564 0.96 TP53 (0.50) NR1H4TP53MEN1KMT2AALDH1A1
SCHEMBL7997469 0.91 NR1H4 (0.52) NR1H4TP53MEN1KMT2A
SCHEMBL8001670 0.91 MEN1 (0.53) NR1H4MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL8002281 0.91 MEN1 (0.53) NR1H4MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL7988822 0.90 TP53 (0.48) NR1H4TP53MEN1KMT2AKDM4E
SCHEMBL7998977 0.88 TP53 (0.46) NR1H4TP53MEN1KMT2AKDM4E
SCHEMBL6579035 0.87 NPC1 (0.46) TP53MEN1KMT2AKDM4EALDH1A1
SCHEMBL8000975 0.85 MEN1 (0.49) NR1H4MEN1KMT2ASMN1; SMN2
SCHEMBL8000665 0.85 MEN1 (0.51) NR1H4MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL7975873 0.84 MAPT (0.52) TP53MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1161337-C Chinolinelone derivative, its prepn. method and antiabnormal reaction agent ���ձ���ī��ѧ��ҵ��ʽ���� 2004-08-11 CN disclosed
CN-1158265-C Quinoline ketone derivant and antianaphylaction using same as active substance ���ձ���ī��ѧ��ҵ��ʽ���� 2004-07-21 CN disclosed
EP-0927718-B1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK & CHEMICALS (JP) 2004-02-25 EP disclosed
CN-1095834-C Quinolinone derivatives and antiallergic agent containing said quinolinone derivatives as active ingredient DAINIPPON INK & CHEMICALS (JP) 2002-12-11 CN disclosed
US-6271416-B1 O-(HYDROCARBONOXYACETAMIDO)BENZOIC ACID DERIVATIVES AS INTERMEDIATES DAINIPPON INK AND CHEMICALS, INC. (JP) 2001-08-07 US disclosed
CN-1275564-A Quinoline ketone derivant and antianaphylaction using same as active substance DAINIPPON INK & CHEMICALS (JP) 2000-12-06 CN disclosed
US-6136822-A ETHER, HYDROXY QUINOLINONE COMPOUNDS DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-10-24 US disclosed
US-6114352-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-09-05 US disclosed
EP-0785190-B1 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK & CHEMICALS (JP) 2000-08-16 EP disclosed
US-5942521-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-08-24 US disclosed
EP-0927718-A1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-07-07 EP disclosed
CN-1221738-A Chinolinelone derivative, its prepn. method and antiabnormal reaction agent DAINIPPON INK & CHEMICALS (JP) 1999-07-07 CN disclosed
CN-1163268-A Quinolinone derivatives and antiallergic agent containing said quinolinone derivatives as active ingredient LAINIPPON INK AND CHEMICALC IN (JP) 1997-10-29 CN disclosed
EP-0785190-A2 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1997-07-23 EP disclosed