SCHEMBL6579858

SCHEMBL6579858

CCOc1c(O)c2ccccc2[nH]c1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 14/20 0.57
ALDH1A1 P00352 9/20 0.57
HPGD P15428 5/20 0.57
MAPT P10636 2/20 0.57
IDE P14735 1/20 0.57
MPI P34949 1/20 0.57
CACNA1B Q00975 1/20 0.57
APBA1 Q02410 1/20 0.57
HSD17B10 Q99714 6/20 0.55
GRIN2D O15399 1/20 0.54
GRIN3B O60391 1/20 0.54
GRIN1 Q05586 1/20 0.54
GRIN2A Q12879 1/20 0.54
GRIN2B Q13224 1/20 0.54
GRIN2C Q14957 1/20 0.54
GRIN3A Q8TCU5 1/20 0.54
GAA P10253 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
DAO P14920 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6579272 0.88 KDM4E (0.59) KDM4EALDH1A1HPGDMAPTIDE
SCHEMBL6577224 0.82 KDM4E (0.66) KDM4EALDH1A1HPGDMAPTIDE
SCHEMBL6579326 0.80 KDM4E (0.50) KDM4EALDH1A1HPGDMAPTIDE
SCHEMBL7116110 0.80 GRIN2D (0.58) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL16651204 0.80 GSK3B (0.47) HPGDMAPTHSD17B10MEN1KMT2A
SCHEMBL6579453 0.78 KDM4E (0.57) KDM4EALDH1A1HPGDMAPTIDE
SCHEMBL9000750 0.76 KDM4E (0.57) KDM4EALDH1A1HPGDMAPTIDE
SCHEMBL10050059 0.76 KDM4E (0.77) KDM4EALDH1A1HPGDMAPTIDE
SCHEMBL9448851 0.75 GAA (0.41) ALDH1A1HPGDMAPTGAAMEN1
SCHEMBL1058188 0.75 KDM5A (0.68) KDM4EALDH1A1HPGDHSD17B10GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927718-B1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK & CHEMICALS (JP) 2004-02-25 EP disclosed
US-6271416-B1 O-(HYDROCARBONOXYACETAMIDO)BENZOIC ACID DERIVATIVES AS INTERMEDIATES DAINIPPON INK AND CHEMICALS, INC. (JP) 2001-08-07 US disclosed
US-6136822-A ETHER, HYDROXY QUINOLINONE COMPOUNDS DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-10-24 US disclosed
US-6114352-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 2000-09-05 US disclosed
EP-0785190-B1 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK & CHEMICALS (JP) 2000-08-16 EP disclosed
US-5942521-A Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-08-24 US disclosed
EP-0927718-A1 Quinolinone derivative, method for preparing the same, and anti-allergic agent DAINIPPON INK AND CHEMICALS, INC. (JP) 1999-07-07 EP disclosed
EP-0785190-A2 Quinolinone derivative and antiallergic agent with said quinolinone derivative as the active ingredient DAINIPPON INK AND CHEMICALS, INC. (JP) 1997-07-23 EP disclosed