SCHEMBL6580723

SCHEMBL6580723

C#CCn1nc(-c2cccc(C=O)c2)nc1-c1ccc(OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 2/20 0.47
NR1H3 Q13133 2/20 0.47
MAOB P27338 5/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
MAOA P21397 1/20 0.40
TSHR P16473 1/20 0.38
AVPR1B P47901 3/20 0.36
TGM2 P21980 1/20 0.36
TGM1 P22735 1/20 0.36
CASP3 P42574 1/20 0.36
TGM3 Q08188 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
MEN1 O00255 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6578570 0.96 MAOB (0.43) NR1H2NR1H3MAOBNPC1RAB9A
SCHEMBL6580724 0.90 NR1H3 (0.47) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6584155 0.87 NR1H3 (0.51) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6578401 0.85 NR1H2 (0.43) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6578548 0.85 NR1H3 (0.64) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6584100 0.84 NR1H2 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6584148 0.84 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6578958 0.84 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6581065 0.84 NR1H3 (0.48) NR1H2NR1H3NPC1RAB9ATDP1
SCHEMBL6581319 0.84 NR1H2 (0.46) NR1H2NR1H3NPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed