SCHEMBL6580914

SCHEMBL6580914

CN(C)Cc1cccc(-c2n[nH]c(-c3ccc(OC(F)F)cc3)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.46
NR1H3 Q13133 5/20 0.46
ADORA2A P29274 2/20 0.42
ADORA1 P30542 2/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ATAD2 Q6PL18 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
S1PR1 P21453 2/20 0.40
BCHE P06276 3/20 0.38
LMNA P02545 1/20 0.37
DGAT1 O75907 1/20 0.37
HTR7 P34969 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6584137 0.99 NR1H2 (0.46) NR1H2NR1H3ADORA2AADORA1NPC1
SCHEMBL6578554 0.86 NR1H2 (0.47) NR1H2NR1H3ADORA2AADORA1NPC1
SCHEMBL6581627 0.85 S1PR1 (0.42) NR1H2NR1H3ADORA2AADORA1NPC1
Hydrochloric Acid SCHEMBL6580524 0.85 NR1H2 (0.58) NR1H2NR1H3ADORA2AADORA1NPC1
Hydrochloric Acid SCHEMBL6578562 0.85 NR1H2 (0.46) NR1H2NR1H3ADORA2AADORA1NPC1
Hydrochloric Acid SCHEMBL6581348 0.85 S1PR1 (0.41) NR1H2NR1H3ADORA2AADORA1NPC1
SCHEMBL27457299 0.84 NPC1 (0.57) NR1H2NR1H3NPC1RAB9AATAD2
Hydrochloric Acid SCHEMBL6578722 0.83 S1PR1 (0.50) NR1H2NR1H3ADORA2AADORA1NPC1
Hydrochloric Acid SCHEMBL6581076 0.82 NPC1 (0.56) NR1H2NR1H3NPC1RAB9AATAD2
Hydrochloric Acid SCHEMBL6581154 0.81 NR1H2 (0.45) NR1H2NR1H3ADORA2AADORA1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP claimed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US claimed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP claimed
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed