SCHEMBL6581315

SCHEMBL6581315

CCOC(=O)Cn1nc(-c2ccc(OC)cc2)nc1-c1cccc(CN(C)C)c1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.59
AVPR1B P47901 15/20 0.46
NR1H2 P55055 1/20 0.44
NR1H3 Q13133 1/20 0.44
MAPT P10636 1/20 0.42
HSD17B2 P37059 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6581313 0.99 TSHR (0.58) TSHRAVPR1BNR1H2NR1H3MAPT
Hydrochloric Acid SCHEMBL6583345 0.95 TSHR (0.58) TSHRAVPR1BNR1H2NR1H3MAPT
Hydrochloric Acid SCHEMBL6578594 0.91 AVPR1B (0.49) TSHRAVPR1BNR1H2NR1H3
Hydrochloric Acid SCHEMBL6580828 0.89 AVPR1B (0.47) TSHRAVPR1BNR1H2NR1H3HSD17B2
Hydrochloric Acid SCHEMBL6578482 0.88 NR1H2 (0.49) TSHRAVPR1BNR1H2NR1H3
Hydrochloric Acid SCHEMBL6581143 0.85 NR1H2 (0.45) AVPR1BNR1H2NR1H3MAPT
SCHEMBL6580598 0.84 NR1H3 (0.47) TSHRAVPR1BNR1H2NR1H3HSD17B2
Hydrochloric Acid SCHEMBL6581513 0.83 NR1H3 (0.46) TSHRAVPR1BNR1H2NR1H3HSD17B2
SCHEMBL7812160 0.83 TSHR (0.62) TSHRAVPR1BMAPT
SCHEMBL6578223 0.83 NR1H2 (0.47) AVPR1BNR1H2NR1H3HSD17B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed