SCHEMBL6582803

SCHEMBL6582803

COc1ccc(-c2nc(-c3cccc(C=O)c3)n(Cc3cccnc3)n2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 4/20 0.51
NR1H2 P55055 3/20 0.51
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.42
GAA P10253 1/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
F2 P00734 3/20 0.41
POLB P06746 1/20 0.41
HSD17B10 Q99714 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
HTT P42858 1/20 0.40
CYP2C9 P11712 2/20 0.39
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6580585 0.96 NR1H3 (0.56) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6582468 0.89 NR1H3 (0.53) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6581539 0.89 NR1H3 (0.64) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6581102 0.89 NR1H3 (0.57) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6582476 0.88 NR1H3 (0.60) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6578522 0.85 NR1H3 (0.59) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6581091 0.85 NR1H3 (0.71) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6578548 0.85 NR1H3 (0.64) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6581357 0.85 NR1H3 (0.53) NR1H3NR1H2ALDH1A1LMNAGAA
SCHEMBL6582807 0.84 NR1H3 (0.66) NR1H3NR1H2ALDH1A1LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1070708-B1 Triazole derivatives HOFFMANN LA ROCHE (CH) 2004-01-14 EP disclosed
US-6265426-B1 CENTRAL NERVOUS SYSTEM DISORDERS HOFFMANN-LA ROCHE INC. 2001-07-24 US disclosed
EP-1070708-A1 Triazole and imidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-01-24 EP disclosed