SCHEMBL6584642

SCHEMBL6584642

O=c1[nH]c2ccccc2n1C1CCCNC1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.61
CHRM4 P08173 2/20 0.61
CHRM1 P11229 2/20 0.61
CHRM3 P20309 1/20 0.61
OPRM1 P35372 11/20 0.53
OPRK1 P41145 7/20 0.53
OPRL1 P41146 7/20 0.53
SLC18A3 Q16572 1/20 0.53
OPRD1 P41143 2/20 0.52
PLD1 Q13393 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
ALDH1A1 P00352 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11203042 0.99 CHRM2 (0.60) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL2636603 0.91 CHRM1 (0.57) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL2636476 0.91 CHRM1 (0.57) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL2636477 0.91 CHRM1 (0.57) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL4084782 0.85 CHRM1 (0.76) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL22605476 0.85 CHRM1 (0.58) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL3142425 0.85 CHRM1 (0.81) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL31285882 0.85 CHRM1 (0.58) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL3146496 0.83 CHRM2 (0.83) CHRM2CHRM4CHRM1CHRM3OPRM1
SCHEMBL15575953 0.83 CHRM2 (0.42) CHRM2CHRM4CHRM1CHRM3OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011513-A1 SHP2 INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND APPLICATION THEREOF 北京泰德制药股份有限公司 2023-02-09 WO disclosed
EP-0990653-B1 2-OXOIMIDAZOLE DERIVATIVES BANYU PHARMA CO LTD (JP) 2004-09-15 EP disclosed
US-6258825-B1 ANALGESIC, A RELIEVER AGAINST TOLERANCE TO A NARCOTIC ANALGESIC REPRESENTED BY MORPHINE, REMEDY FOR PARKINSONISM, A REMEDY FOR CHOREA, AN ANTIDEPRESSANT, A REMEDY FOR DIABETES INSIPIDUS, A REMEDY FOR POLYURIA, OR HYPOTENSION BANYU PHARMACEUTICAL CO., LTD. (JP) 2001-07-10 US disclosed
EP-0990653-A1 2-OXOIMIDAZOLE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 2000-04-05 EP disclosed